SCHEMBL17552183

SCHEMBL17552183

O=C(Nc1cccc2cccnc12)c1ccc(F)cc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.77
KDR P35968 5/20 0.76
L3MBTL1 Q9Y468 2/20 0.75
GAA P10253 2/20 0.75
TDP1 Q9NUW8 1/20 0.75
MAPT P10636 5/20 0.70
TP53 P04637 2/20 0.70
KMT2A Q03164 3/20 0.67
HTT P42858 1/20 0.67
POLB P06746 1/20 0.67
RAB9A P51151 3/20 0.66
NPC1 O15118 2/20 0.66
CASP3 P42574 1/20 0.66
SENP8 Q96LD8 1/20 0.66
SENP7 Q9BQF6 1/20 0.66
SENP6 Q9GZR1 1/20 0.66
KDM4E B2RXH2 2/20 0.65
MEN1 O00255 2/20 0.64
TNKS O95271 2/20 0.64
TNKS2 Q9H2K2 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911198 1.00 HDAC6 (0.77) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL19631488 0.87 HDAC6 (1.00) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL15270551 0.87 HDAC6 (0.79) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL29647754 0.87 HDAC6 (1.00) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL6260903 0.87 KDR (1.00) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL29434873 0.87 KDR (1.00) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL19422867 0.86 KDR (0.72) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL19748451 0.86 HDAC6 (0.73) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL29911021 0.86 KDR (0.72) HDAC6KDRL3MBTL1GAATDP1
SCHEMBL29655108 0.86 HDAC6 (0.73) HDAC6KDRL3MBTL1GAATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2024-01-18 US disclosed
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-11-28 US disclosed
EP-4037685-B1 QUINOLINE THAT MODULATE SERCA AND ITS USE FOR TREATING DISEASE NEURODON CORP (US) 2023-09-20 EP disclosed
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2023-09-14 US disclosed
CN-116744928-A Quinolines modulating SERCA and their use for treating diseases 神经元公司 2023-09-12 CN disclosed
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-08-22 US disclosed
CN-113336784-B 3-substituted benzofluorenone or 3-substituted naphthofluorenone derivatives and synthesis method thereof 上海大学 2022-11-18 CN disclosed
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2022-01-20 US disclosed
CN-113336784-A 3-substituted benzofluorenone or 3-substituted naphthofluorenone derivatives and synthesis method thereof 上海大学 2021-09-03 CN disclosed
CN-111575731-B Method for electrochemically synthesizing C5 and C7 dihalogenated quinoline amide derivatives 浙江工业大学 2021-08-24 CN disclosed
US-10772881-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION 2020-09-15 US disclosed
CN-111575731-A Method for electrochemically synthesizing C5 and C7 dihalogenated quinoline amide derivatives 浙江工业大学 2020-08-25 CN disclosed
CN-109320497-B Method for preparing phenanthridinone compound by copper compound induction 广州大学 2020-07-31 CN disclosed
CN-106938985-B 5-site alkenylated 8-acylaminoquinoline compound and one-pot preparation method thereof 湖南大学 2020-05-05 CN disclosed
CN-107698586-B Method for preparing pyridoquinazolinone compound by catalysis of copper compound 广州大学 2020-02-07 CN disclosed
US-20190151303-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2019-05-23 US disclosed
CN-109320497-A A method of phenanthridines ketone compounds are prepared by copper compound induction 广州大学 2019-02-12 CN disclosed
CN-107698586-A It is a kind of that the method for preparing Pyridine-quinazolinocompound compound is catalyzed by copper compound 广州大学 2018-02-16 CN disclosed
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES EIGER BIOPHARMACEUTICALS, INC. (US) 2017-10-05 US disclosed
WO-2016032569-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES CELLADON CORPORATION (US) 2016-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 HDAC6 1539/4885KDR 4506/4885L3MBTL1 4692/4885
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES ATP2A1, ATP2A3, ATP2A2 HDAC6 611/4885KDR 4844/4885L3MBTL1 3273/4885
US-10772881-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 HDAC6 1841/4885KDR 4683/4885L3MBTL1 4561/4885
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 HDAC6 1539/4885KDR 4506/4885L3MBTL1 4692/4885
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 HDAC6 1539/4885KDR 4506/4885L3MBTL1 4692/4885
US-20190151303-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 HDAC6 1841/4885KDR 4683/4885L3MBTL1 4561/4885
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 HDAC6 1539/4885KDR 4506/4885L3MBTL1 4692/4885
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 HDAC6 1539/4885KDR 4506/4885L3MBTL1 4692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.