SCHEMBL17552185

SCHEMBL17552185

Cc1ccc2cccc(NC(=O)c3cccc(OC(F)(F)F)c3)c2n1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.67
POLB P06746 1/20 0.67
MAPT P10636 3/20 0.52
GAA P10253 1/20 0.52
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
TSHR P16473 1/20 0.52
HSD17B10 Q99714 1/20 0.52
ALOX12 P18054 1/20 0.52
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
MCHR1 Q99705 1/20 0.48
KAT6A Q92794 1/20 0.48
THRB P10828 1/20 0.48
GRM5 P41594 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911228 1.00 TP53 (0.67) TP53POLBMAPTGAAALDH1A1
SCHEMBL17540883 0.89 MAPT (0.58) TP53POLBMAPTGAAALDH1A1
SCHEMBL17552237 0.84 TP53 (0.70) TP53POLBMAPTGAAALDH1A1
SCHEMBL29911115 0.84 TP53 (0.70) TP53POLBMAPTGAAALDH1A1
SCHEMBL1035541 0.84 KAT6A (0.48) TP53POLBALDH1A1MEN1KMT2A
SCHEMBL17552192 0.83 GAA (0.64) TP53POLBMAPTGAAALDH1A1
SCHEMBL29911165 0.83 GAA (0.64) TP53POLBMAPTGAAALDH1A1
SCHEMBL17552190 0.81 POLB (0.62) TP53POLBMAPTGAAALDH1A1
SCHEMBL29911073 0.81 POLB (0.62) TP53POLBMAPTGAAALDH1A1
SCHEMBL26798522 0.81 NPC1 (0.72) TP53POLBMAPTGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2024-01-18 US disclosed
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-11-28 US disclosed
EP-4037685-B1 QUINOLINE THAT MODULATE SERCA AND ITS USE FOR TREATING DISEASE NEURODON CORP (US) 2023-09-20 EP disclosed
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2023-09-14 US disclosed
CN-116744928-A Quinolines modulating SERCA and their use for treating diseases 神经元公司 2023-09-12 CN disclosed
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-08-22 US disclosed
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2022-01-20 US disclosed
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2020-11-05 US disclosed
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES EIGER BIOPHARMACEUTICALS, INC. (US) 2017-10-05 US disclosed
WO-2016032569-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES CELLADON CORPORATION (US) 2016-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230285382-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES ATP2A1, ATP2A3, ATP2A2 TP53 3254/4885POLB 2994/4885MAPT 1538/4885
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 TP53 3732/4885POLB 3166/4885MAPT 1228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.