SCHEMBL17552192

SCHEMBL17552192

Cc1ccc2cccc(NC(=O)c3cccc(C(F)(F)F)c3)c2n1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.64
TP53 P04637 1/20 0.59
POLB P06746 1/20 0.59
PTGS1 P23219 1/20 0.57
ALDH1A1 P00352 3/20 0.55
MAPT P10636 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ALOX12 P18054 1/20 0.55
BRAF P15056 2/20 0.54
RAB9A P51151 2/20 0.54
HTT P42858 1/20 0.54
KCNK3 O14649 1/20 0.53
KCNK9 Q9NPC2 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
CSF1R P07333 1/20 0.53
KIT P10721 1/20 0.53
P2RX1 P51575 1/20 0.52
LMNA P02545 1/20 0.52
NPC1 O15118 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29911165 1.00 GAA (0.64) GAATP53POLBPTGS1ALDH1A1
SCHEMBL17540885 0.89 MAPT (0.58) GAATP53POLBPTGS1ALDH1A1
SCHEMBL29911073 0.84 POLB (0.62) GAATP53POLBALDH1A1MAPT
SCHEMBL17552190 0.84 POLB (0.62) GAATP53POLBALDH1A1MAPT
SCHEMBL26798522 0.84 NPC1 (0.72) GAATP53POLBALDH1A1MAPT
SCHEMBL28249147 0.83 RAB9A (0.67) GAATP53PTGS1ALDH1A1MAPT
SCHEMBL30733198 0.83 RAB9A (0.67) GAATP53PTGS1ALDH1A1MAPT
SCHEMBL17552185 0.83 TP53 (0.67) GAATP53POLBALDH1A1MAPT
SCHEMBL29911228 0.83 TP53 (0.67) GAATP53POLBALDH1A1MAPT
SCHEMBL28154257 0.82 MAPT (0.76) GAATP53POLBALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2024-01-18 US disclosed
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-11-28 US disclosed
EP-4037685-B1 QUINOLINE THAT MODULATE SERCA AND ITS USE FOR TREATING DISEASE NEURODON CORP (US) 2023-09-20 EP disclosed
CN-116744928-A Quinolines modulating SERCA and their use for treating diseases 神经元公司 2023-09-12 CN disclosed
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION (US) 2023-08-22 US disclosed
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2022-01-20 US disclosed
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2020-11-05 US disclosed
US-10772881-B2 Quinolines that modulate SERCA and their use for treating disease NEURODON CORPORATION 2020-09-15 US disclosed
US-20190151303-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE NEURODON CORPORATION 2019-05-23 US disclosed
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES EIGER BIOPHARMACEUTICALS, INC. (US) 2017-10-05 US disclosed
WO-2016032569-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES CELLADON CORPORATION (US) 2016-03-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170281611-A1 QUINOLINES AND THEIR USE FOR TREATING ENDOPLASMIC RETICULUM STRESS-CAUSED DISEASES ATP2A1, ATP2A3, ATP2A2 GAA 36/4885TP53 3254/4885POLB 2994/4885
US-10772881-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 GAA 65/4885TP53 3639/4885POLB 3596/4885
US-11730729-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 GAA 94/4885TP53 3732/4885POLB 3166/4885
US-11827626-B2 Quinolines that modulate SERCA and their use for treating disease ATP2A1, ATP2A3, ATP2A2 GAA 94/4885TP53 3732/4885POLB 3166/4885
US-20190151303-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 GAA 65/4885TP53 3639/4885POLB 3596/4885
US-20220016108-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 GAA 94/4885TP53 3732/4885POLB 3166/4885
US-20200347038-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 GAA 94/4885TP53 3732/4885POLB 3166/4885
US-20240016793-A1 QUINOLINES THAT MODULATE SERCA AND THEIR USE FOR TREATING DISEASE ATP2A1, ATP2A3, ATP2A2 GAA 94/4885TP53 3732/4885POLB 3166/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.