SCHEMBL1755233

SCHEMBL1755233

CN/C=C\Nc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 7/20 0.46
HPGD P15428 6/20 0.46
TSHR P16473 3/20 0.46
HSD17B10 Q99714 3/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
ALOX15 P16050 1/20 0.46
CDC25B P30305 1/20 0.46
ATM Q13315 1/20 0.46
KDM4E B2RXH2 6/20 0.43
GAA P10253 3/20 0.43
MAPT P10636 3/20 0.42
CA12 O43570 3/20 0.42
CA14 Q9ULX7 3/20 0.42
CA4 P22748 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
CA3 P07451 1/20 0.42
CA6 P23280 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6696812 0.78 KDM4E (0.48) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL1342156 0.78 ALDH1A1 (0.50) KEAP1ALDH1A1HPGDTSHRHSD17B10
Hydrochloric Acid SCHEMBL3159285 0.77 ALDH1A1 (0.49) KEAP1ALDH1A1HPGDTSHRHSD17B10
Hydrochloric Acid SCHEMBL27946264 0.77 ALDH1A1 (0.49) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL4652710 0.76 TSHR (0.48) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL20715566 0.76 ALDH1A1 (0.44) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL49308 0.74 KEAP1 (0.61) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL1755252 0.74 KEAP1 (0.43) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL4632499 0.74 ALDH1A1 (0.47) KEAP1ALDH1A1HPGDTSHRHSD17B10
SCHEMBL4632503 0.74 ALDH1A1 (0.47) KEAP1ALDH1A1HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569919-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2012-04-18 EP disclosed
US-7642277-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-05 US disclosed