SCHEMBL1755253

SCHEMBL1755253

O=C(CSc1nccn1-c1cccc2ccccc12)Nc1ccccc1[N+](=O)[O-]

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.65
LMNA P02545 5/20 0.59
MAPT P10636 4/20 0.58
HPGD P15428 1/20 0.57
THRB P10828 1/20 0.56
ALDH1A1 P00352 7/20 0.53
CYP1A2 P05177 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
CYP2C19 P33261 1/20 0.51
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MAPK1 P28482 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
POLB P06746 1/20 0.48
NPC1 O15118 1/20 0.48
TSHR P16473 1/20 0.47
KDM4E B2RXH2 1/20 0.47
APOBEC3A P31941 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1702862 0.85 ALDH1A1 (0.56) TP53LMNAMAPTALDH1A1CYP1A2
SCHEMBL1702962 0.81 ALDH1A1 (0.66) LMNAMAPTHPGDALDH1A1CYP1A2
SCHEMBL13236226 0.75 TP53 (1.00) TP53LMNAMAPTHPGDTHRB
SCHEMBL1702876 0.70 MAPT (0.52) TP53LMNAMAPTHPGDALDH1A1
SCHEMBL1703004 0.69 ALDH1A1 (0.52) LMNAMAPTALDH1A1CYP1A2L3MBTL1
SCHEMBL6403512 0.69 KMT2A (0.70) LMNAMAPTALDH1A1CYP1A2MEN1
SCHEMBL4207071 0.68 PTGES (0.72) LMNAALDH1A1CYP1A2L3MBTL1MEN1
SCHEMBL5821874 0.67 ALDH1A1 (0.53) LMNAMAPTALDH1A1CYP1A2L3MBTL1
SCHEMBL6277594 0.67 ALDH1A1 (0.64) LMNAMAPTHPGDALDH1A1CYP1A2
SCHEMBL4207324 0.67 ALDH1A1 (0.62) TP53LMNAMAPTHPGDTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569919-B1 NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2012-04-18 EP disclosed
US-7642277-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-05 US disclosed
US-7642277-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-01-05 US disclosed