SCHEMBL17558356

SCHEMBL17558356

CNC(=O)c1cc(C(C)C2(C(C)c3ccnc(C(=O)NC)c3)NC(=O)N(c3ccc(SC(F)(F)F)cc3)C2=O)ccn1

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IGF1R P08069 12/20 0.56
PDE2A O00408 8/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174717 0.90 IGF1R (0.54) IGF1RPDE2A
SCHEMBL6174941 0.90 IGF1R (0.45) IGF1RPDE2A
SCHEMBL6174371 0.85 IGF1R (0.44) IGF1RPDE2A
SCHEMBL6176345 0.85 IGF1R (0.53) IGF1R
SCHEMBL6173555 0.84 IGF1R (0.41) IGF1RPDE2A
SCHEMBL6175683 0.84 IGF1R (0.51) IGF1R
SCHEMBL6174494 0.84 IGF1R (0.42) IGF1R
SCHEMBL6172820 0.84 IGF1R (0.42) IGF1R
SCHEMBL17558385 0.84 IGF1R (0.56) IGF1R
SCHEMBL6173419 0.84 IGF1R (0.42) IGF1RPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3188729-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS Genzyme Corporation (US) 2017-07-12 EP disclosed
WO-2016036796-A1 CYCLIC UREA COMPOUNDS AS TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS GENZYME CORPORATION (US) 2016-03-10 WO disclosed