SCHEMBL17568804

SCHEMBL17568804

CC(C)CC1(C)NC(=N)N(CC2CCCN(Sc3ccccc3)C2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.33
GFER P55789 1/20 0.32
ABCB11 O95342 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
ADRA2A P08913 1/20 0.31
CHRM1 P11229 1/20 0.31
ADRA2B P18089 1/20 0.31
CHRM3 P20309 1/20 0.31
DRD1 P21728 1/20 0.31
PTGS1 P23219 1/20 0.31
SLC6A2 P23975 1/20 0.31
ADRA1D P25100 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
ADRA1A P35348 1/20 0.31
HRH1 P35367 1/20 0.31
OPRM1 P35372 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17568795 0.86 SMN1; SMN2 (0.32) SMN1; SMN2ALDH1A1GAAL3MBTL1
SCHEMBL17568791 0.82 ABCB11 (0.37) SMN1; SMN2GFERABCB11CHRM2CHRM4
SCHEMBL7526022 0.81 CYP2C19 (0.39) SMN1; SMN2LMNA
SCHEMBL7521580 0.81 ALDH1A1 (0.40) SMN1; SMN2GFERALDH1A1L3MBTL1LMNA
SCHEMBL7520457 0.81 GRM5 (0.39) SMN1; SMN2GFERALDH1A1LMNAADAMTS5
SCHEMBL7527996 0.80 CPB1 (0.40) SMN1; SMN2GFERALDH1A1ADAMTS5
SCHEMBL12593309 0.80 CPB1 (0.40) SMN1; SMN2GFERALDH1A1ADAMTS5
SCHEMBL7526060 0.80 ALDH1A1 (0.41) SMN1; SMN2ALDH1A1LMNA
SCHEMBL7521707 0.80 TACR3 (0.43) SMN1; SMN2ALDH1A1GAAL3MBTL1LMNA
SCHEMBL7518635 0.79 HPGD (0.48) SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2153832-B1 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS MERCK SHARP & DOHME (US) 2016-03-09 EP disclosed