SCHEMBL17586283

SCHEMBL17586283

CN(C(=O)OC(C)(C)C)C12CC(C(C)(C)C)(C1)C2

nearest known ligand 0.31

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ASGR1 P07306 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17586288 0.87 HDAC6 (0.32) ASGR1HDAC1HDAC2HDAC6
SCHEMBL17582445 0.85 ASGR1 (0.33) ASGR1
SCHEMBL17586292 0.82 ASGR1 (0.32) ASGR1HDAC1HDAC2HDAC6
SCHEMBL23284466 0.81 ASGR1 (0.31) ASGR1HDAC1HDAC2HDAC6
SCHEMBL30885816 0.79 ASGR1 (0.31) ASGR1HDAC1HDAC2HDAC6
SCHEMBL18038888 0.79 ASGR1 (0.31) ASGR1HDAC1HDAC2HDAC6
SCHEMBL24462299 0.79 ASGR1 (0.31) ASGR1HDAC1HDAC2HDAC6
SCHEMBL20848346 0.78 ASGR1 (0.38) ASGR1HDAC1HDAC2HDAC6
SCHEMBL17586268 0.78 OPRM1 (0.32)
SCHEMBL20848339 0.77 DGAT1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10975035-B2 Bicyclic compounds RECURIUM IP HOLDINGS, LLC (US) 2021-04-13 US disclosed
US-20190233377-A1 BICYCLIC COMPOUNDS Zeno Royalties & Milestones, LLC 2019-08-01 US disclosed
US-10308609-B2 Bicyclic compounds Zeno Royalties & Milestones, LLC (US) 2019-06-04 US disclosed
US-20160075654-A1 BICYCLIC COMPOUNDS RECURIUM IP HOLDINGS, LLC 2016-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190233377-A1 BICYCLIC COMPOUNDS OPRK1, OPRM1, OPRL1 ASGR1 4577/4885HDAC1 486/4885HDAC2 487/4885
US-20160075654-A1 BICYCLIC COMPOUNDS OPRK1, OPRM1, OPRL1 ASGR1 4577/4885HDAC1 486/4885HDAC2 487/4885
US-10975035-B2 Bicyclic compounds OPRK1, OPRM1, OPRL1 ASGR1 4577/4885HDAC1 486/4885HDAC2 487/4885
US-10308609-B2 Bicyclic compounds OPRK1, OPRM1, OPRL1 ASGR1 4577/4885HDAC1 486/4885HDAC2 487/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.