SCHEMBL1758656

SCHEMBL1758656

O=C(Cc1ccc(CCCC23CC4CC(CC(C4)C2)C3)cc1)NO

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 7/20 0.49
HDAC1 Q13547 6/20 0.49
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
HDAC6 Q9UBN7 4/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
P2RX7 Q99572 1/20 0.42
EPHX2 P34913 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758576 0.96 HDAC1 (0.51) HDAC8HDAC1NPC1RAB9AHDAC6
SCHEMBL1758604 0.84 HDAC6 (0.59) HDAC6MEN1KMT2AEPHX2
SCHEMBL1758674 0.84 HDAC6 (0.52) HDAC8HDAC1RAB9AHDAC6MEN1
SCHEMBL6878384 0.82 HDAC1 (0.44) HDAC8HDAC1HDAC6MEN1KMT2A
SCHEMBL1758695 0.80 MEP1B (0.46) HDAC8HDAC1RAB9AHDAC6MEN1
SCHEMBL15522678 0.77 HDAC1 (0.74) HDAC8HDAC1HDAC6MEN1KMT2A
SCHEMBL1759196 0.74 MEN1 (0.52) NPC1RAB9AHDAC6MEN1KMT2A
SCHEMBL28060952 0.74 EPHX2 (0.57) NPC1RAB9AMEN1KMT2AP2RX7
SCHEMBL4658066 0.73 CNR2 (0.58) P2RX7EPHX2
SCHEMBL1758784 0.73 NPC1 (0.48) HDAC8NPC1RAB9AHDAC6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed