SCHEMBL1758604

SCHEMBL1758604

O=C(Cc1ccc(OCCCC23CC4CC(CC(C4)C2)C3)cc1)NO

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.59
KDM4E B2RXH2 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2D6 P10635 1/20 0.59
PDE4A P27815 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
HIF1A Q16665 1/20 0.59
HDAC10 Q969S8 1/20 0.59
ALDH1A1 P00352 2/20 0.48
EPHX2 P34913 5/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LMNA P02545 1/20 0.42
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880270 0.87 HDAC6 (0.50) HDAC6KDM4ECYP1A2CYP2D6PDE4A
SCHEMBL1758656 0.84 HDAC8 (0.49) HDAC6EPHX2MEN1KMT2A
SCHEMBL1758576 0.83 HDAC1 (0.51) HDAC6HDAC10MEN1KMT2A
SCHEMBL1758674 0.80 HDAC6 (0.52) HDAC6SMN1; SMN2HDAC10EPHX2MEN1
SCHEMBL2749026 0.78 EPHX2 (0.63) ALDH1A1EPHX2MEN1KMT2ALMNA
SCHEMBL1758671 0.78 ALDH1A1 (0.60) HDAC6KDM4ECYP1A2CYP2D6PDE4A
SCHEMBL1758860 0.77 HDAC6 (0.58) HDAC6KDM4ECYP1A2CYP2D6PDE4A
SCHEMBL1758695 0.76 MEP1B (0.46) HDAC6ALDH1A1EPHX2MEN1KMT2A
Bufexamac SCHEMBL25215 0.75 KDM4E (1.00) HDAC6KDM4ECYP1A2CYP2D6PDE4A
Bufexamac SCHEMBL5076113 0.75 KDM4E (1.00) HDAC6KDM4ECYP1A2CYP2D6PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed