SCHEMBL1758680

SCHEMBL1758680

CC(N(C(=O)O)c1nc(CC(=O)NO)cs1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.42
HDAC6 Q9UBN7 3/20 0.41
PDE5A O76074 10/20 0.39
KDM4E B2RXH2 2/20 0.39
PDE1A P54750 2/20 0.36
PDE1B Q01064 2/20 0.36
PDE1C Q14123 2/20 0.36
SHMT1 P34896 2/20 0.35
SHMT2 P34897 2/20 0.35
GAA P10253 2/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758697 0.79 PDE5A (0.40) HDAC6PDE5AKDM4EPDE1APDE1B
SCHEMBL1758679 0.77 PDE5A (0.41) HDAC6PDE5AKDM4EPDE1APDE1B
SCHEMBL1758935 0.77 PDE5A (0.39) ALDH1A1PDE5AKDM4EPDE1APDE1B
SCHEMBL1758740 0.75 PDE5A (0.37) HDAC6PDE5AKDM4EPDE1APDE1B
SCHEMBL1758936 0.71 MAPT (0.38) ALDH1A1HDAC6PDE5AKDM4EPDE1A
SCHEMBL1758659 0.70 PDE5A (0.38) ALDH1A1PDE5AKDM4EPDE1APDE1B
SCHEMBL1759205 0.68 CNR2 (0.62) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758713 0.67 PDE5A (0.54) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758649 0.66 EPHX2 (0.63) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758672 0.65 HDAC1 (0.41) HDAC6PDE5AKDM4EPDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed