SCHEMBL1758686

SCHEMBL1758686

O=C(NO)C(F)(F)c1csc(CC23CC4CC(CC(C4)C2)C3)n1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 5/20 0.34
CNR2 P34972 1/20 0.33
GLA P06280 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC8 Q9BY41 2/20 0.32
EPHX2 P34913 3/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
P2RX7 Q99572 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758655 0.75 CNR2 (0.59) CNR2KMT2AEPHX2GAANPC1
SCHEMBL6879978 0.64 CNR2 (0.45) HDAC6CNR2HDAC8EPHX2GAA
SCHEMBL1758648 0.62 CNR2 (0.60) CNR2KMT2AEPHX2GAANPC1
SCHEMBL1758672 0.60 HDAC1 (0.41) HDAC6HDAC8
SCHEMBL6384681 0.56 ALDH1A1 (0.61) EPHX2P2RX7
SCHEMBL4907174 0.56 MEN1 (0.34) KMT2AGAAPOLBRAB9A
SCHEMBL31532570 0.55 IDH1 (0.32)
SCHEMBL22570461 0.55 ALDH1A1 (0.68) GLAKMT2AEPHX2P2RX7
SCHEMBL23547606 0.55 NPSR1 (0.44) KMT2AHPGDNPC1RAB9A
SCHEMBL24917625 0.55 HDAC3 (0.35) HDAC6HDAC8GAANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed