SCHEMBL1758692

SCHEMBL1758692

O=C(Cc1csc(NC(=O)CCc2ccc(C34CC5CC(CC(C5)C3)C4)cc2)n1)NO

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 15/20 0.56
PDE1A P54750 6/20 0.56
PDE1B Q01064 6/20 0.56
PDE1C Q14123 6/20 0.56
KDM4E B2RXH2 2/20 0.47
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878814 0.82 PDE5A (0.49) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1759219 0.79 HDAC3 (0.55) GAAHTTLMNA
SCHEMBL1759205 0.79 CNR2 (0.62) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758601 0.79 PDE5A (0.54) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758713 0.78 PDE5A (0.54) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758880 0.77 PDE5A (0.41) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1759195 0.76 GAA (0.53) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758817 0.75 PDE5A (0.50) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758649 0.75 EPHX2 (0.63) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758738 0.72 PDE5A (0.48) PDE5APDE1APDE1BPDE1CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed