SCHEMBL1758880

SCHEMBL1758880

O=C(Cc1csc(N(CCCc2ccc(C34CC5CC(CC(C5)C3)C4)cc2)C(=O)O)n1)NO

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 5/20 0.41
PDE1A P54750 2/20 0.41
PDE1B Q01064 2/20 0.41
PDE1C Q14123 2/20 0.41
KDM4E B2RXH2 1/20 0.35
HDAC6 Q9UBN7 4/20 0.34
HDAC1 Q13547 3/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CASP2 P42575 1/20 0.34
LMNA P02545 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758740 0.82 PDE5A (0.37) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758679 0.80 PDE5A (0.41) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758697 0.78 PDE5A (0.40) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758692 0.77 PDE5A (0.56) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758703 0.77 PDE5A (0.40) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758935 0.76 PDE5A (0.39) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758659 0.74 PDE5A (0.38) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758680 0.70 ALDH1A1 (0.42) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758784 0.68 NPC1 (0.48) HDAC6NPC1RAB9ACASP2LMNA
SCHEMBL3604375 0.67 PDE5A (0.44) PDE5APDE1APDE1BPDE1CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed