SCHEMBL1758860

SCHEMBL1758860

O=C(Cc1ccc(OCCCCC2C3CC4CC(C3)CC2C4)cc1)NO

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.58
HDAC10 Q969S8 2/20 0.58
KDM4E B2RXH2 1/20 0.58
CYP1A2 P05177 1/20 0.58
CYP2D6 P10635 1/20 0.58
PDE4A P27815 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
HIF1A Q16665 1/20 0.58
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
MMP3 P08254 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880970 0.88 KDM4E (0.55) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL1758604 0.77 HDAC6 (0.59) HDAC6HDAC10KDM4ECYP1A2CYP2D6
Bufexamac SCHEMBL5076113 0.74 KDM4E (1.00) HDAC6HDAC10KDM4ECYP1A2CYP2D6
Bufexamac SCHEMBL25215 0.74 KDM4E (1.00) HDAC6HDAC10KDM4ECYP1A2CYP2D6
Bufexamac SCHEMBL15456779 0.73 KDM4E (0.97) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL6880270 0.72 HDAC6 (0.50) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL2777642 0.71 CYP1A2 (0.88) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL4580666 0.71 HDAC6 (0.71) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL11296680 0.71 HDAC6 (0.71) HDAC6HDAC10KDM4ECYP1A2CYP2D6
SCHEMBL12688087 0.71 HDAC6 (0.67) HDAC6HDAC10KDM4ECYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed