SCHEMBL17592016

SCHEMBL17592016

Cn1cc(-c2cc3c(-c4nc5cccnc5[nH]4)n[nH]c3cn2)cn1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 15/20 0.65
PIM3 Q86V86 3/20 0.64
PIM2 Q9P1W9 3/20 0.64
CLK2 P49760 3/20 0.59
CLK3 P49761 3/20 0.59
DYRK1A Q13627 3/20 0.59
WNT1 P04628 2/20 0.59
TGFBR1 P36897 1/20 0.57
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17566753 0.88 PIM1 (0.71) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17593591 0.87 AXL (0.59) CLK2CLK3DYRK1AWNT1
SCHEMBL17568376 0.85 PIM1 (0.66) PIM1PIM3PIM2CLK2CLK3
SCHEMBL18474541 0.84 CLK2 (0.53) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17592391 0.83 WNT1 (0.66) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17555578 0.83 CLK2 (0.80) PIM1PIM3PIM2CLK2CLK3
SCHEMBL18440826 0.83 CLK2 (0.70) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17564774 0.83 CLK2 (0.53) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17592351 0.82 PIM1 (0.68) PIM1PIM3PIM2CLK2CLK3
SCHEMBL17592115 0.82 WNT1 (0.64) PIM1PIM3PIM2CLK2CLK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016040184-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF SAMUMED, LLC (US) 2016-03-17 WO claimed
US-20180201624-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2018-07-19 US disclosed
US-20180201624-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2018-07-19 US disclosed
US-9815854-B2 3-(3H-imidazo[4,5-B]pyridin-2-yl)-1H-pyrazolo[3,4-C]pyridine and therapeutic uses thereof SAMUMED, LLC (US) 2017-11-14 US disclosed
US-9815854-B2 3-(3H-imidazo[4,5-B]pyridin-2-yl)-1H-pyrazolo[3,4-C]pyridine and therapeutic uses thereof SAMUMED, LLC (US) 2017-11-14 US disclosed
US-20170260209-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2017-09-14 US disclosed
US-20170260209-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2017-09-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180201624-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF WNT3, WNT1, WNT3A PIM1 1804/4885PIM3 996/4885PIM2 1918/4885
US-20170260209-A1 3-(3H-IMIDAZO[4,5-B]PYRIDIN-2-YL)-1H-PYRAZOLO[3,4-C]PYRIDINE AND THERAPEUTIC USES THEREOF WNT3, WNT1, WNT3A PIM1 1804/4885PIM3 996/4885PIM2 1918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.