SCHEMBL17595028

SCHEMBL17595028

CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(-n2cccc2)cc1.CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(N2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
ALK Q9UM73 1/20 0.42
GPR119 Q8TDV5 3/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
NAMPT P43490 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
HTT P42858 2/20 0.40
ESR2 Q92731 1/20 0.40
NPC1 O15118 1/20 0.40
NR2F2 P24468 1/20 0.40
KIT P10721 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ESRRB O95718 1/20 0.39
ESR1 P03372 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14745432 0.94 MAPT (0.47) ALDH1A1LMNAMAPTALKGPR119
SCHEMBL17595032 0.92 LMNA (0.42) ALDH1A1LMNAMAPTALKGPR119
SCHEMBL14745604 0.84 POLB (0.43) ALDH1A1LMNAMEN1KMT2A
SCHEMBL17595141 0.81 ABCB1 (0.40) ALDH1A1LMNAMAPTALKGPR119
SCHEMBL14745621 0.81 L3MBTL1 (0.43) ALDH1A1LMNAMAPTGPR119SMN1; SMN2
SCHEMBL14741099 0.79 PARP1 (0.41) ALDH1A1LMNAMAPTHTT
SCHEMBL14745092 0.79 PARP1 (0.43) ALDH1A1LMNAMAPTSMN1; SMN2HTT
SCHEMBL14741042 0.78 DHODH (0.44) ALDH1A1LMNAMAPTSMN1; SMN2HTT
SCHEMBL14745094 0.78 PDE3B (0.40) ALDH1A1MAPTSMN1; SMN2CYP2C19
SCHEMBL14740829 0.77 SLC16A3 (0.45) ALDH1A1LMNAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed