SCHEMBL176019

SCHEMBL176019

C=CCC1=NCCc2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.54
ALDH1A1 P00352 2/20 0.54
NOS3 P29474 2/20 0.49
NOS2 P35228 1/20 0.49
MAOA P21397 1/20 0.41
ADRA1D P25100 2/20 0.39
ADRA1A P35348 2/20 0.39
ADRA1B P35368 1/20 0.39
CES1 P23141 1/20 0.38
SLC6A2 P23975 2/20 0.35
SLC22A1 O15245 1/20 0.35
CACNA1F O60840 1/20 0.35
NTRK1 P04629 1/20 0.35
CYP1A2 P05177 1/20 0.35
ADRB2 P07550 1/20 0.35
RET P07949 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
ADRB1 P08588 1/20 0.35
HTR1A P08908 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757777 1.00 KDM4E (0.54) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL20356526 0.82 TSHR (0.44) KDM4EALDH1A1NOS3NOS2ADRA1D
SCHEMBL7819962 0.80 KDM4E (0.58) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL29361631 0.78 KDM4E (0.60) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL7509399 0.78 KDM4E (0.60) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL22995932 0.77 KDM4E (0.63) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL9815282 0.77 ALDH1A1 (0.58) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL30952113 0.77 KDM4E (0.63) KDM4EALDH1A1NOS3NOS2MAOA
Hydrochloric Acid SCHEMBL3452241 0.75 KDM4E (0.57) KDM4EALDH1A1NOS3NOS2MAOA
SCHEMBL24224408 0.74 NOS3 (0.55) KDM4EALDH1A1NOS3NOS2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114874139-B Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2024-02-06 CN claimed
CN-114874139-A Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2022-08-09 CN claimed
CN-114874139-B Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2024-02-06 CN disclosed
CN-114874139-B Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2024-02-06 CN disclosed
CN-114874139-B Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2024-02-06 CN disclosed
CN-114874139-A Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2022-08-09 CN disclosed
CN-114874139-A Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2022-08-09 CN disclosed
CN-114874139-A Synthesis method of 1-benzyl or allyl 3, 4-dihydroisoquinoline 新疆大学 2022-08-09 CN disclosed
EP-2611788-B1 NICOTINE COMPOUNDS AND ANALOGS THEREOF, SYNTHETIC METHODS OF MAKING COMPOUNDS, AND METHODS OF USE UNIV FLORIDA (US) 2017-04-12 EP disclosed
US-9440948-B2 Nicotine compounds and analogs thereof, synthetic methods of making compounds, and methods of use UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2016-09-13 US disclosed
EP-2611788-A2 NICOTINE COMPOUNDS AND ANALOGS THEREOF, SYNTHETIC METHODS OF MAKING COMPOUNDS, AND METHODS OF USE University of Florida Research Foundation, Incorporated (US) 2013-07-10 EP disclosed
US-6277861-B1 FOR TREATMENT AND PROPHYLAXIS OF NERVOUS SYSTEM DISORDERS, PSYCHOLOGICAL DISORDERS, MUSCULAR DISORDERS, DRUG ADDICTION WITHDRAWAL, PAIN SMITHKLINE BEECHAM, P.L.C. (GB) 2001-08-21 US disclosed
EP-1104404-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2001-06-06 EP disclosed
WO-2000009486-A1 SUBSTITUTED ISOQUINOLINE DERIVATIVES AND THEIR USE AS ANTICONVULSIVANTS SMITHKLINE BEECHAM P.L.C. (GB) 2000-02-24 WO disclosed
EP-0971897-A1 ANTI-CONVULSANT ISOQUINOLYL-BENZAMIDE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 2000-01-19 EP disclosed
WO-1998041507-A1 ANTI-CONVULSANT ISOQUINOLYL-BENZAMIDE DERIVATIVES SMITHKLINE BEECHAM PLC (GB) 1998-09-24 WO disclosed
US-4766217-A Preparation of 5,6-dihydro-pyrrolo[2,1-a]isoquinolines BOEHRINGER INGELHEIM KG (DE) 1988-08-23 US disclosed
EP-0150474-B1 Process for the preparation of 5,6-dihydro-pyrrolo-[2,1-a]isoquinolines BOEHRINGER INGELHEIM KG (DE) 1988-08-17 EP disclosed
US-4694085-A CHEMICAL INTERMEDIATES BOEHRINGER INGELHEIM KG (DE) 1987-09-15 US disclosed
EP-0150474-A2 Process for the preparation of 5,6-dihydro-pyrrolo-[2,1-a]isoquinolines BOEHRINGER INGELHEIM KG (DE) 1985-08-07 EP disclosed