SCHEMBL17604686

SCHEMBL17604686

NNC(=O)c1ccc2c(c1)COB2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 2/20 0.41
CYP3A4 P08684 2/20 0.41
BLM P54132 2/20 0.41
KDM5A P29375 1/20 0.41
GFER P55789 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
ALDH1A1 P00352 8/20 0.40
KDM4E B2RXH2 6/20 0.40
MAPT P10636 6/20 0.40
LMNA P02545 4/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
OGG1 O15527 1/20 0.40
SMN1; SMN2 Q16637 4/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TP53 P04637 1/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17604630 0.88 MPO (0.41) MPOCYP3A4BLMKDM5AGFER
SCHEMBL17604678 0.75 KDM4E (0.46) ALDH1A1KDM4EMAPTSMN1; SMN2NPC1
SCHEMBL17620525 0.71 ALDH1A1 (0.57) MPOCYP3A4BLMKDM5AGFER
SCHEMBL20481887 0.69 TSHR (0.42) ALDH1A1KDM4E
SCHEMBL6582556 0.68 NPC1 (0.62) MPOCYP3A4BLMKDM5AGFER
SCHEMBL19608153 0.67 CA12 (0.46) BLMALDH1A1KDM4EMAPTL3MBTL1
SCHEMBL17604604 0.67 MPO (0.39) MPOCYP3A4BLMKDM5AGFER
SCHEMBL17604681 0.67 MAPT (0.39) MPOCYP3A4BLMKDM5AGFER
SCHEMBL17604649 0.67 MPO (0.39) MPOCYP3A4BLMKDM5AGFER
SCHEMBL1395940 0.67 TAS1R3 (0.63) KDM4ESMN1; SMN2NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3194359-A1 BORON-CONTAINING DIACYLHYDRAZINE COMPOUNDS Intrexon Corporation (US) 2017-07-26 EP claimed
WO-2016044390-A1 BORON-CONTAINING DIACYLHYDRAZINE COMPOUNDS INTREXON CORPORATION (US) 2016-03-24 WO claimed