SCHEMBL17607355

SCHEMBL17607355

CC(C)(C)OC(=O)N(CC=CC(=O)O)CCCc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 9/20 0.43
HDAC3 O15379 1/20 0.40
HDAC4 P56524 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
CYP3A4 P08684 2/20 0.39
CHRNA7 P36544 2/20 0.39
NAMPT P43490 1/20 0.39
RIPK1 Q13546 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PTAFR P25105 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17623484 0.83 TBXAS1 (0.51) TBXAS1CYP3A4CHRNA7RIPK1TDP1
SCHEMBL17623481 0.82 TBXAS1 (0.56) TBXAS1CYP3A4CHRNA7TDP1L3MBTL1
SCHEMBL17607353 0.79 TBXAS1 (0.40) TBXAS1CYP3A4NAMPTRIPK1L3MBTL1
SCHEMBL17623485 0.78 TBXAS1 (0.47) TBXAS1CYP3A4CHRNA7RIPK1TDP1
SCHEMBL4289433 0.77 L3MBTL1 (0.44) HDAC3HDAC1HDAC2L3MBTL1
SCHEMBL17623600 0.76 TBXAS1 (0.45) TBXAS1CYP3A4CHRNA7TDP1L3MBTL1
SCHEMBL30154236 0.75 CA14 (0.40) HDAC3HDAC1HDAC2HDAC6
SCHEMBL17607354 0.75 TBXAS1 (0.42) TBXAS1CYP3A4CHRNA7TDP1L3MBTL1
SCHEMBL17623497 0.74 TBXAS1 (0.43) TBXAS1HDAC3HDAC4HDAC1HDAC7
SCHEMBL17623499 0.74 TBXAS1 (0.43) TBXAS1CYP3A4CHRNA7TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016042280-A1 CONJUGATES OF AMINO ACID-PYRIDINE/PYRIDINIUM AND USES THEREOF AS BIOCIDAL AGENTS Université de Nice Sophia Antipolis (FR) 2016-03-24 WO disclosed