SCHEMBL17619985

SCHEMBL17619985

FC(F)(F)c1ccc(-c2cnccn2)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.47
MAPT P10636 1/20 0.44
KCNH2 Q12809 3/20 0.43
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
PIK3CA P42336 3/20 0.41
PI4KB Q9UBF8 3/20 0.41
MAP4K4 O95819 1/20 0.41
MINK1 Q8N4C8 1/20 0.41
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
PIK3CD O00329 2/20 0.40
PIK3CB P42338 2/20 0.40
PI4KA P42356 2/20 0.40
PIK3CG P48736 2/20 0.40
WNT3A P56704 1/20 0.40
TRPV3 Q8NET8 1/20 0.39
PIM1 P11309 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30527142 0.80 CYP2A6 (0.50) TRPV4
SCHEMBL17247906 0.80 CYP2A6 (0.50) TRPV4
SCHEMBL2858005 0.79 KIF11 (0.55) CYP2D6CYP19A1CYP2C9CYP2C19ABL1
SCHEMBL28863764 0.79 ABL1 (0.48) TRPV4MAPTKCNH2CYP2D6PIK3CA
SCHEMBL30636554 0.78 CYP2A6 (0.56) TRPV4
SCHEMBL11541937 0.77 CYP2D6 (0.60) MAPTCYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL20224611 0.77 CYP2D6 (0.38) MAPTCYP2D6CYP19A1CYP2C9CYP2C19
SCHEMBL17247907 0.76 CYP2A6 (0.53) TRPV4KCNH2PIK3CAPI4KBMAP4K4
SCHEMBL28242951 0.76 TRPV4 (0.42) TRPV4KCNH2CYP2C19PIK3CAPI4KB
SCHEMBL28021874 0.75 KCNH2 (0.50) TRPV4KCNH2PIK3CAPI4KBMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104869997-B novel compounds as diacylglycerol acyltransferase inhibitors 葛兰素史密斯克莱有限责任公司 2017-03-22 CN disclosed
WO-2016044792-A1 INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL HYDRA BIOSCIENCES, INC. (US) 2016-03-24 WO disclosed