SCHEMBL17620896

SCHEMBL17620896

COc1cccc(OC)c1CNC(N)=Nc1ccc2ccccc2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.45
MEN1 O00255 3/20 0.45
NOD2 Q9HC29 1/20 0.42
ADORA2A P29274 1/20 0.41
ALDH1A1 P00352 4/20 0.40
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
KDM4E B2RXH2 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
PKM P14618 1/20 0.39
CNR2 P34972 1/20 0.39
HPGD P15428 3/20 0.38
MAPT P10636 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
NFKB1 P19838 1/20 0.36
HTT P42858 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4629836 0.88 KMT2A (0.59) KMT2AMEN1NOD2ALDH1A1NPC1
SCHEMBL2782915 0.82 MEN1 (0.44) KMT2AMEN1NOD2ADORA2AALDH1A1
SCHEMBL2782723 0.81 ADORA2A (0.39) KMT2AADORA2AALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL2780729 0.80 PLAU (0.50) ALDH1A1NPC1RAB9AKDM4ESMN1; SMN2
SCHEMBL2782184 0.80 AGTR1 (0.39) KMT2AMEN1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL2780662 0.79 ADRA2A (0.53) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL2777876 0.78 SMN1; SMN2 (0.48) KMT2AMEN1ALDH1A1NPC1RAB9A
SCHEMBL2380137 0.78 ROCK2 (0.39) KMT2AMEN1ALDH1A1MAPTGAA
SCHEMBL2780849 0.77 ADRA2A (0.50) KMT2AMEN1ADORA2AALDH1A1NPC1
SCHEMBL2779998 0.77 ROCK2 (0.42) KMT2AMEN1ALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9296697-B2 Hetaryl-substituted guanidine compounds and use thereof as binding partners for 5-HT5-receptors ABBOTT LABORATORIES (US) 2016-03-29 US claimed