SCHEMBL17643003

SCHEMBL17643003

O=c1c2cc(Br)ccc2nc(-c2ccccc2)n1-c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.68
KMT2A Q03164 6/20 0.68
ATM Q13315 1/20 0.68
GAA P10253 2/20 0.61
MAPT P10636 3/20 0.57
HSP90AA1 P07900 1/20 0.57
ALDH1A1 P00352 6/20 0.53
AVPR1A P37288 1/20 0.53
LMNA P02545 1/20 0.53
HTT P42858 2/20 0.52
HCAR1 Q9BXC0 1/20 0.51
KDM4E B2RXH2 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17643006 0.92 MEN1 (0.59) MEN1KMT2AATMGAAMAPT
SCHEMBL15810554 0.87 KMT2A (0.56) MEN1KMT2AATMGAAMAPT
SCHEMBL17643200 0.85 MEN1 (0.62) MEN1KMT2AATMGAAMAPT
SCHEMBL17642998 0.85 MEN1 (0.68) MEN1KMT2AGAAMAPTHSP90AA1
SCHEMBL17643007 0.84 MEN1 (0.70) MEN1KMT2AGAAMAPTHSP90AA1
SCHEMBL17629396 0.84 MEN1 (0.70) MEN1KMT2AGAAMAPTHSP90AA1
SCHEMBL17642999 0.83 MEN1 (0.66) MEN1KMT2AGAAMAPTHSP90AA1
SCHEMBL21658056 0.83 MEN1 (0.65) MEN1KMT2AATMGAAMAPT
SCHEMBL14571460 0.82 KMT2A (0.80) MEN1KMT2AGAAMAPTHSP90AA1
SCHEMBL9953980 0.81 ATM (0.51) MEN1KMT2AATMMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3197982-B1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2020-05-06 EP disclosed
US-10544360-B2 Materials for organic electroluminescent devices MERCK PATENT GMBH (DE) 2020-01-28 US disclosed
WO-2016045765-A1 MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES MERCK PATENT GMBH (DE) 2016-03-31 WO disclosed