SCHEMBL17656221

SCHEMBL17656221

CCc1ccc2c(c1)NC(=O)c1ccc(C)cc1N2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1G1 Q9HCP0 1/20 0.61
ROS1 P08922 1/20 0.53
CDK5 Q00535 1/20 0.53
ACVR1 Q04771 1/20 0.53
LRRK2 Q5S007 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 2/20 0.48
NPC1 O15118 1/20 0.48
CYP1A2 P05177 1/20 0.48
MAPT P10636 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
RAB9A P51151 1/20 0.48
MCL1 Q07820 1/20 0.48
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
CHEK1 O14757 10/20 0.45
HSD17B10 Q99714 1/20 0.44
TGM2 P21980 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14985677 0.87 CSNK1G1 (0.77) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL5327486 0.79 MAOA (0.63) SMN1; SMN2ALDH1A1NPC1MAPTRAB9A
SCHEMBL23242561 0.79 ALDH1A1 (0.49) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL14985676 0.77 ACVR1 (0.83) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL18462586 0.77 ACVR1 (0.83) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL9980151 0.77 CSNK1G1 (0.61) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL2756590 0.77 CSNK1G1 (0.61) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL9185276 0.76 CSNK1G1 (1.00) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL17656324 0.74 SMN1; SMN2 (0.46) CSNK1G1ROS1CDK5ACVR1LRRK2
SCHEMBL12124081 0.73 SMN1; SMN2 (0.47) SMN1; SMN2ALDH1A1GAANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-A1 ANTIVIRAL COMPOUNDS Gilead Pharmasset LLC (US) 2016-04-06 EP disclosed