SCHEMBL17698019

SCHEMBL17698019

COC(C)c1cc(NC(=O)c2ccc(C(C)(C)C)cc2)ccc1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 12/20 0.54
PPARG P37231 5/20 0.53
PPARA Q07869 4/20 0.53
KCNK9 Q9NPC2 1/20 0.52
TP53 P04637 2/20 0.52
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
PPARD Q03181 1/20 0.50
GPBAR1 Q8TDU6 1/20 0.50
HDAC3 O15379 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
LMNA P02545 1/20 0.48
KCNK3 O14649 1/20 0.48
TRPV1 Q8NER1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17698020 0.76 NR1H4 (0.57) NR1H4PPARGPPARAKCNK9TP53
SCHEMBL7297239 0.73 NR1H4 (0.81) NR1H4KCNK9SMN1; SMN2HDAC3HDAC11
SCHEMBL3873116 0.73 NR1H4 (0.81) NR1H4KCNK9SMN1; SMN2HDAC3HDAC11
SCHEMBL7303163 0.72 HDAC3 (0.86) NR1H4MAPTSMN1; SMN2HDAC3HDAC11
SCHEMBL5697470 0.71 NR1H4 (0.68) NR1H4TP53MAPTSMN1; SMN2HDAC3
SCHEMBL9696412 0.71 NR1H4 (0.77) NR1H4PPARGPPARAKCNK9TP53
SCHEMBL4611487 0.70 HDAC3 (0.71) NR1H4TP53MAPTSMN1; SMN2HDAC3
SCHEMBL3882727 0.70 HDAC3 (0.71) NR1H4TP53MAPTSMN1; SMN2HDAC3
SCHEMBL557111 0.70 HDAC6 (0.71) NR1H4KCNK9TP53MAPTSMN1; SMN2
SCHEMBL7301440 0.70 SMN1; SMN2 (0.78) NR1H4TP53MAPTSMN1; SMN2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2716285-B9 Compounds for treating and/or preventing diseases associated with bone loss CENTRE NAT DE LA RECH SCIENT -CNRS- (FR) 2017-03-01 EP claimed
EP-2716285-B1 Compounds for treating and/or preventing diseases associated with bone loss CENTRE NAT RECH SCIENT (FR) 2016-04-27 EP claimed