SCHEMBL17706151

SCHEMBL17706151

Cc1ccc(SN2CCNC(=O)C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
CRBN Q96SW2 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
DDB1 Q16531 1/20 0.36
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
GFER P55789 1/20 0.35
RAB9A P51151 3/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 2/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 2/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTR1A P08908 2/20 0.33
HTR3A P46098 2/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19381879 0.79 MAPT (0.41) CRBNSMN1; SMN2RAB9AALDH1A1NPC1
SCHEMBL19986858 0.75 ADRB1 (0.52) RAB9AALDH1A1NPC1KDM4EHTR1A
SCHEMBL10999156 0.71 ADRB1 (0.56) ALOX5SMN1; SMN2TOP2ATOP2BMAPT
SCHEMBL21009009 0.71
SCHEMBL18583232 0.69 HPGD (0.43) SMN1; SMN2RAB9AALDH1A1NPC1PKM
SCHEMBL20627373 0.69 L3MBTL1 (0.35) ALOX5TOP2ATOP2BGFERRAB9A
SCHEMBL17468364 0.68 CXCR4 (0.55) SMN1; SMN2ALDH1A1KDM4EGAAPOLB
SCHEMBL15196278 0.68 L3MBTL1 (0.37) ALOX5SMN1; SMN2TOP2ATOP2BGFER
SCHEMBL3928664 0.68 GFER (0.69) SMN1; SMN2GFERALDH1A1PKMGAA
SCHEMBL19563446 0.67 HPGD (0.34) SMN1; SMN2RAB9AALDH1A1NPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3012250-A1 ISOQUINOLINE MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2016-04-27 EP disclosed