SCHEMBL1773253

SCHEMBL1773253

CC(C)(C)OC(=O)N1CCC(CC#N)C1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
MAPT P10636 1/20 0.56
KMT2A Q03164 1/20 0.56
NR1H2 P55055 1/20 0.46
HPGD P15428 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PKM P14618 1/20 0.44
CTSK P43235 1/20 0.43
GPR119 Q8TDV5 5/20 0.43
RECQL P46063 1/20 0.43
EPHX1 P07099 1/20 0.43
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41
USP2 O75604 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FAAH O00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15626875 1.00 MEN1 (0.56) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL15626878 1.00 MEN1 (0.56) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL13542527 0.92 MEN1 (0.64) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL12940814 0.92 MEN1 (0.64) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL11995200 0.92 MEN1 (0.64) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL123942 0.91 MEN1 (0.52) MEN1ALDH1A1MAPTKMT2AHPGD
SCHEMBL31420572 0.90 MEN1 (0.60) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL31421174 0.90 MEN1 (0.60) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL9696880 0.88 NR1H2 (0.54) MEN1ALDH1A1MAPTKMT2ANR1H2
SCHEMBL16162498 0.87 MEN1 (0.48) MEN1ALDH1A1MAPTKMT2ANR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166117-B Heteroaromatic compounds as VANIN inhibitors 勃林格殷格翰国际公司 2025-04-15 CN disclosed
EP-3475286-B1 SUBSTITUTED PYRROLO [2, 3-D]PYRIDAZIN-4-ONES AND PYRAZOLO [3, 4-D]PYRIDAZIN-4-ONES AS PROTEIN KINASE INHIBITORS FOCHON PHARMACEUTICALS LTD (CN) 2025-03-26 EP disclosed
CN-113226462-B Heteroaromatic compounds as VANIN inhibitors 勃林格殷格翰国际公司 2025-02-11 CN disclosed
CN-116018138-A Substituted 1H-imidazo [1,2-b ] pyrazole-3-carboxamides as inhibitors of brunauer tyrosine kinase 河南知微生物医药有限公司 2023-04-25 CN disclosed
US-20230081390-A1 INHIBITORS OF RAF KINASES Pierre Fabre Médicament (FR) 2023-03-16 US disclosed
WO-2022012550-A1 SUBSTITUTED 1H-IMIDAZO [1, 2-B] PYRAZOLE-3-CARBOXAMIDE AS BRUTON'S TYROSINE KINASE INHIBITORS HENAN NORMAL UNIVERSITY (CN) 2022-01-20 WO disclosed
CN-113874381-A Inhibitors of RAF kinase 金耐特生物制药公司 2021-12-31 CN disclosed
CN-109476666-B Compound as kinase inhibitor 上海复尚慧创医药研究有限公司 2021-10-15 CN disclosed
CN-113226462-A Heteroaromatic compounds as VANIN inhibitors 勃林格殷格翰国际公司 2021-08-06 CN disclosed
CN-113166117-A Heteroaromatic compounds as VANIN inhibitors 勃林格殷格翰国际公司 2021-07-23 CN disclosed
CN-109476666-A Substituted pyrrolo [2,3-d ] pyridazin-4-ones and pyrazolo [3,4-d ] pyridazin-4-ones as kinase inhibitors 上海复尚慧创医药研究有限公司 2019-03-15 CN disclosed
US-10023561-B2 Fumagillol heterocyclic compounds and methods of making and using same ZAFGEN, INC. (US) 2018-07-17 US disclosed
EP-3334728-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME Zafgen, Inc. (US) 2018-06-20 EP disclosed
US-20170342058-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. 2017-11-30 US disclosed
US-9682965-B2 Fumagillol heterocyclic compounds and methods of making and using same ZAFGEN, INC. (US) 2017-06-20 US disclosed
US-20170066749-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. 2017-03-09 US disclosed
WO-2017027684-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN, INC. (US) 2017-02-16 WO disclosed
EP-2705030-B1 PARTIALLY SATURATED TRICYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME ZAFGEN INC (US) 2016-07-27 EP disclosed
US-20110112103-A1 5-HYDROXYPYRIMIDINE-4-CARBOXAMIDE COMPOUND DAIICHI SANKYO COMPANY, LIMITED (JP) 2011-05-12 US disclosed
WO-1992002521-A1 1-AZABICYCLO[3.2.0]HEPT-2-ENE-2-CARBOXYLIC ACID COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170066749-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME METAP2, FAP, FOLH1 MEN1 350/4885ALDH1A1 450/4885MAPT 1422/4885
US-20170342058-A1 FUMAGILLOL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING SAME METAP2, FAP, FOLH1 MEN1 350/4885ALDH1A1 450/4885MAPT 1422/4885
US-20230081390-A1 INHIBITORS OF RAF KINASES BRAF, RAF1, ARAF MEN1 2171/4885ALDH1A1 2750/4885MAPT 2859/4885
US-10023561-B2 Fumagillol heterocyclic compounds and methods of making and using same METAP2, FAP, FOLH1 MEN1 350/4885ALDH1A1 450/4885MAPT 1422/4885
US-20110112103-A1 5-HYDROXYPYRIMIDINE-4-CARBOXAMIDE COMPOUND EPOR, CBR1, CBR3 MEN1 2513/4885ALDH1A1 1179/4885MAPT 4845/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.