SCHEMBL17733488

SCHEMBL17733488

CSc1ccc2c(c1)C=CCC2

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
HTR7 P34969 1/20 0.34
TYMS P04818 1/20 0.31
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30205863 0.85 HTR2A (0.32) HTR2AHTR2CHTR2BHTR7MCL1
SCHEMBL27677971 0.81 HTR7 (0.39) HTR2AHTR2CHTR2BHTR7TYMS
SCHEMBL29501037 0.75 PARP10 (0.34)
SCHEMBL9114452 0.75 PARP10 (0.34)
SCHEMBL25675742 0.72 ANPEP (0.31)
SCHEMBL29634842 0.71 PNMT (0.37) HTR2AHTR2CHTR2B
SCHEMBL31503035 0.71 CA9 (0.35)
SCHEMBL2524442 0.71
SCHEMBL30344009 0.71 KDM1A (0.37) HTR2AHTR2C
SCHEMBL7650098 0.71 CA9 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110072864-A TDO2 INHIBITORS 基因泰克公司 2019-07-30 CN disclosed
EP-1696912-B1 PYRAZOLOPYRIDINES AND ANALOGS THEREOF 3M INNOVATIVE PROPERTIES CO (US) 2016-05-11 EP disclosed