SCHEMBL1773993

SCHEMBL1773993

CC1(C)C(=O)N(c2ccc(Oc3ccc(Cl)cc3)cc2)C(=O)N1Cc1ccccc1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.42
SMO Q99835 2/20 0.41
IGF1R P08069 4/20 0.39
TAS2R8 Q9NYW2 2/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
ELANE P08246 2/20 0.37
HTR2A P28223 1/20 0.37
SLC6A4 P31645 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PPARG P37231 1/20 0.36
PPARD Q03181 1/20 0.36
PPARA Q07869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12603131 0.94 AR (0.43) ARIGF1RTAS2R8PPARGPPARD
SCHEMBL8034783 0.94 SMO (0.45) ARSMOIGF1RTAS2R8ELANE
SCHEMBL8029468 0.87 ELANE (0.44) ARIGF1RTAS2R8ELANE
SCHEMBL1773362 0.87 PPARG (0.51) ARIGF1RTAS2R8PPARGPPARD
SCHEMBL1772428 0.86 AR (0.54) AR
SCHEMBL12603120 0.85 IGF1R (0.44) ARIGF1RTAS2R8ELANEPPARG
SCHEMBL8030958 0.85 ELANE (0.46) ARIGF1RTAS2R8ELANE
SCHEMBL12603179 0.85 LMNA (0.44) ARIGF1RTAS2R8LMNA
SCHEMBL12603129 0.85 MCHR1 (0.42) ARIGF1RTAS2R8LMNA
SCHEMBL8029780 0.85 NPC1 (0.43) ARIGF1RTAS2R8SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
WO-2009097997-A1 SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof GIPR, PGC, DDC AR 2449/4885SMO 3229/4885IGF1R 189/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.