SCHEMBL1774235

SCHEMBL1774235

CC1(C)NC(=O)N(c2ccc(S(=O)(=O)N3CCOCC3)cc2)C1=O

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 5/20 0.52
KDM4E B2RXH2 2/20 0.52
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PKM P14618 1/20 0.48
ALDH1A1 P00352 4/20 0.48
GAA P10253 2/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
USP2 O75604 1/20 0.47
HSD17B10 Q99714 1/20 0.47
AR P10275 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
PHOSPHO1 Q8TCT1 1/20 0.46
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1772860 0.87 LMNA (0.57) POLBKDM4ELMNASMN1; SMN2GAA
SCHEMBL5177701 0.82 AR (0.55) POLBKDM4ESMN1; SMN2ALDH1A1MEN1
SCHEMBL12793245 0.75 POLB (0.88) POLBKDM4ELMNASMN1; SMN2ALDH1A1
SCHEMBL1772437 0.75 AR (0.57) POLBLMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL12793319 0.73 LMNA (0.73) POLBKDM4ELMNASMN1; SMN2ALDH1A1
SCHEMBL1773397 0.72 AR (0.54) POLBLMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL4028165 0.71 AR (0.53) POLBLMNASMN1; SMN2MEN1KMT2A
SCHEMBL12793723 0.71 POLB (0.73) POLBKDM4ELMNASMN1; SMN2ALDH1A1
SCHEMBL171151 0.71 POLB (0.73) POLBKDM4ELMNASMN1; SMN2PKM
SCHEMBL10306750 0.71 POLB (0.73) POLBKDM4ELMNASMN1; SMN2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
EP-2242747-A1 SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF Sanofi-Aventis (FR) 2010-10-27 EP disclosed
WO-2009097997-A1 SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof GIPR, PGC, DDC POLB 3357/4885KDM4E 585/4885LMNA 1453/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.