SCHEMBL177559

SCHEMBL177559

NC(=O)CCCS(=O)(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.55
BLM P54132 4/20 0.46
CYP2C19 P33261 3/20 0.46
LMNA P02545 2/20 0.46
SLC6A6 P31641 1/20 0.46
PTGS1 P23219 1/20 0.39
PDE4A P27815 1/20 0.39
KMT2A Q03164 2/20 0.32
TP53 P04637 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 2/20 0.32
MEN1 O00255 1/20 0.32
FAAH O00519 1/20 0.32
SOAT1 P35610 1/20 0.32
ALOX15 P16050 2/20 0.32
PMP22 Q01453 2/20 0.32
APEX1 P27695 1/20 0.32
KDM4E B2RXH2 2/20 0.32
GMNN O75496 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177764 0.97 APP (0.52) APPBLMCYP2C19LMNASLC6A6
SCHEMBL177845 0.97 APP (0.52) APPBLMCYP2C19LMNASLC6A6
SCHEMBL8592959 0.92 APP (0.52) APPBLMCYP2C19LMNASLC6A6
SCHEMBL20902773 0.90 APP (0.50) APPBLMCYP2C19LMNASLC6A6
SCHEMBL19569862 0.90 APP (0.50) APPBLMCYP2C19LMNASLC6A6
SCHEMBL9702032 0.90 APP (0.50) APPBLMCYP2C19LMNASLC6A6
SCHEMBL177492 0.86
SCHEMBL177593 0.83 BLM (0.46) APPBLMCYP2C19LMNASLC6A6
SCHEMBL177490 0.83 BLM (0.46) APPBLMCYP2C19LMNASLC6A6
SCHEMBL29045770 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694505-B1 HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2022-04-27 EP claimed
US-10201623-B2 HSP90-targeted cardiac imaging and therapy MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2019-02-12 US claimed
US-20140088121-A1 HSP90 Inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2014-03-27 US claimed
US-20240058482-A1 USES OF LABELED HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2024-02-22 US disclosed
US-11661398-B2 Cellular transport system for transferring a sulfonic acid construct carrying a cargo into the cytoplasm of a cell Scientist of Fortune, S.A. (LU) 2023-05-30 US disclosed
US-11607465-B2 Uses of labeled HSP90 inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2023-03-21 US disclosed
CN-109071454-B Sulfonylureas and related compounds and uses thereof 昆士兰大学 2023-02-17 CN disclosed
EP-2694505-B1 HSP90 INHIBITORS SLOAN KETTERING INST CANCER RES (US) 2022-04-27 EP disclosed
CN-109374889-B Use of labeled HSP90 inhibitors 索隆-基特林癌症研究协会 2022-04-19 CN disclosed
CN-113521314-A HSP 90-Targeted inflammation and infection imaging and treatment 纪念斯隆-凯特琳癌症中心 2021-10-22 CN disclosed
US-20210308285-A1 HSP90-TARGETED INFLAMMATION AND INFECTION IMAGING AND THERAPY MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2021-10-07 US disclosed
US-5338815-A Used in thickeners, dispersion stabilizers and lubricants SHOWA DENKO K.K. (JP) 1994-08-16 US disclosed
US-5300606-A Crosslinked N-vinylamide resin SHOWA DENKO K.K. (JP) 1994-04-05 US disclosed
US-5280095-A N-vinylcarboxylic acid amine resin SHOWA DENKO K.K. (JP) 1994-01-18 US disclosed
EP-0510246-A1 Use of fine particulate crosslinked type n-vinylamide resin microgel SHOWA DENKO KABUSHIKI KAISHA (JP) 1992-10-28 EP disclosed
EP-0473881-A1 Liquid absorption agent SHOWA DENKO KABUSHIKI KAISHA (JP) 1992-03-11 EP disclosed
EP-0215124-B1 SILVER HALIDE PHOTOGRAPHIC PHOTO-SENSITIVE MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1991-09-04 EP disclosed
US-4925782-A Silver halide photographic light-sensitive element containing water soluble dye compounds FUJI PHOTO FILM CO., LTD. (JP) 1990-05-15 US disclosed
US-4879204-A HIGH CONTRAST FUJI PHOTO FILM CO., LTD. (JP) 1989-11-07 US disclosed
EP-0215124-A1 SILVER HALIDE PHOTOGRAPHIC PHOTO-SENSITIVE MATERIAL FUJI PHOTO FILM CO., LTD. (JP) 1987-03-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11661398-B2 Cellular transport system for transferring a sulfonic acid construct carrying a cargo into the cytoplasm of a cell GOT1, GGCT, TGM2 APP 4021/4885BLM 3378/4885CYP2C19 3074/4885
US-20140088121-A1 HSP90 Inhibitors HSP90AB1, HSP90B1, HSP90AB2P APP 3963/4885BLM 1490/4885CYP2C19 558/4885
US-20240058482-A1 USES OF LABELED HSP90 INHIBITORS HSP90AB1, HSP90B1, HSP90AA1 APP 4713/4885BLM 2589/4885CYP2C19 3730/4885
US-10201623-B2 HSP90-targeted cardiac imaging and therapy HSP90AB1, HSP90AA1, HSP90B1 APP 3551/4885BLM 3028/4885CYP2C19 1829/4885
US-11607465-B2 Uses of labeled HSP90 inhibitors HSP90AB1, HSP90B1, HSP90AA1 APP 4713/4885BLM 2589/4885CYP2C19 3730/4885
US-20210308285-A1 HSP90-TARGETED INFLAMMATION AND INFECTION IMAGING AND THERAPY HSP90AB1, HSP90AA1, HSP90B1 APP 1633/4885BLM 3846/4885CYP2C19 2183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.