SCHEMBL1776648

SCHEMBL1776648

Cc1onc(-c2ccccc2)c1COc1ccc(C(=O)NC2CCOCC2)nn1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA5 P08648 3/20 0.83
GABRA1 P14867 13/20 0.80
GABRA5 P31644 4/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776448 0.94 GABRA1 (0.78) ITGA5GABRA1GABRA5
SCHEMBL1776675 0.92 ITGA5 (0.81) ITGA5GABRA1GABRA5
SCHEMBL1776643 0.91 GABRA1 (0.80) ITGA5GABRA1GABRA5
SCHEMBL20241323 0.91 ITGA5 (1.00) ITGA5GABRA1GABRA5
SCHEMBL30592846 0.91 ITGA5 (1.00) ITGA5GABRA1GABRA5
SCHEMBL1777844 0.90 GABRA5 (0.77) ITGA5GABRA1GABRA5
Alogabat SCHEMBL20241000 0.89 GABRA1 (1.00) ITGA5GABRA1
Alogabat SCHEMBL29500971 0.89 GABRA1 (1.00) ITGA5GABRA1
SCHEMBL1777497 0.89 ITGA5 (1.00) ITGA5GABRA1GABRA5
SCHEMBL20241011 0.87 GABRA1 (1.00) ITGA5GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US claimed
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US disclosed