SCHEMBL1777013

SCHEMBL1777013

Cc1onc(-c2ccncn2)c1COc1ccc(C(=O)OCC(N)=O)nn1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 9/20 0.59
GABRA1 P14867 8/20 0.54
ITGA5 P08648 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776679 0.91 GABRA5 (0.63) GABRA5GABRA1ITGA5
SCHEMBL1776363 0.89 GABRA1 (0.60) GABRA5GABRA1ITGA5
SCHEMBL1776592 0.88 ITGA5 (0.61) GABRA5GABRA1ITGA5
SCHEMBL1776663 0.86 GABRA5 (0.63) GABRA5GABRA1ITGA5
SCHEMBL1779475 0.84 GABRA1 (0.61) GABRA5GABRA1
SCHEMBL1776773 0.81 GABRA5 (0.76) GABRA5GABRA1ITGA5
SCHEMBL1778273 0.79 GABRA5 (0.61) GABRA5GABRA1
SCHEMBL1776628 0.79 GABRA1 (0.58) GABRA5GABRA1ITGA5
SCHEMBL1777284 0.79 GABRA5 (0.75) GABRA5GABRA1ITGA5
SCHEMBL1776329 0.78 ITGA5 (0.65) GABRA5GABRA1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US disclosed