SCHEMBL1779475

SCHEMBL1779475

Cc1onc(-c2ccccc2)c1COc1ccc(C(=O)OCC(N)=O)nn1

nearest known ligand 0.61

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 4/20 0.61
GABRA5 P31644 16/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1776363 0.91 GABRA1 (0.60) GABRA1GABRA5
SCHEMBL1777918 0.90 GABRA5 (0.71) GABRA1GABRA5
SCHEMBL1778273 0.89 GABRA5 (0.61) GABRA1GABRA5
SCHEMBL2928471 0.89 GABRA1 (0.76) GABRA1GABRA5
SCHEMBL1776592 0.89 ITGA5 (0.61) GABRA1GABRA5
SCHEMBL108079 0.88 GABRA5 (0.70) GABRA1GABRA5
SCHEMBL107284 0.86 GABRA1 (0.62) GABRA1GABRA5
SCHEMBL286529 0.84 GABRA5 (0.54) GABRA5
SCHEMBL287532 0.84 GABRA5 (0.52) GABRA5
SCHEMBL1777013 0.84 GABRA5 (0.59) GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943619-B2 Isoxazolo-pyridazine derivatives HOFFMANN-LA ROCHE INC. (US) 2011-05-17 US disclosed