SCHEMBL17777985

SCHEMBL17777985

Cc1ccc(Sc2ccccc2Nc2ccccc2N)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.49
GAA P10253 2/20 0.49
MAPT P10636 2/20 0.49
SLC6A4 P31645 10/20 0.44
SLC6A3 Q01959 6/20 0.44
SLC6A2 P23975 6/20 0.44
HTR1A P08908 6/20 0.44
HTR3A P46098 6/20 0.44
CYP1A2 P05177 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 3/20 0.43
ADRB2 P07550 2/20 0.43
ADRB1 P08588 2/20 0.43
CYP3A4 P08684 2/20 0.43
HRH2 P25021 2/20 0.43
HTR1B P28222 2/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
HTR7 P34969 2/20 0.43
HRH1 P35367 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723181 0.82 SLC6A4 (0.57) TDP1MAPTSLC6A4SLC6A3SLC6A2
SCHEMBL29773377 0.82 SLC6A4 (0.57) TDP1MAPTSLC6A4SLC6A3SLC6A2
SCHEMBL30338359 0.82 SLC6A4 (0.57) TDP1MAPTSLC6A4SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL16151212 0.81 SLC6A4 (0.55) TDP1SLC6A4SLC6A3SLC6A2HTR1A
Hydrochloric Acid SCHEMBL30695614 0.81 SLC6A4 (0.55) TDP1SLC6A4SLC6A3SLC6A2HTR1A
SCHEMBL17553862 0.78 HTR1A (0.48) TDP1MAPTSLC6A4SLC6A3SLC6A2
SCHEMBL13057071 0.75 HTR1A (0.57) TDP1GAAMAPTSLC6A4SLC6A3
SCHEMBL14723137 0.75 L3MBTL1 (0.52) TDP1MAPTSLC6A4HTR1AHTR3A
SCHEMBL17777979 0.73 KMT2A (0.57) TDP1MAPTSLC6A4HTR1AHTR3A
SCHEMBL17777986 0.73 HTR1A (0.44) TDP1MAPTSLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016079751-A2 A PROCESS FOR PREPARATION OF VORTIOXETINE AND POLYMORPHS THEREOF MEGAFINE PHARMA (P) LTD. (IN) 2016-05-26 WO disclosed