SCHEMBL17778583

SCHEMBL17778583

CC1(C)OC[C@H](CCOc2ccnc(N)c2)O1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.41
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
CCNK O75909 1/20 0.37
CDK12 Q9NYV4 1/20 0.37
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
CASP1 P29466 1/20 0.35
BLM P54132 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17777000 1.00 MAPK14 (0.41) MAPK14NOS3NOS1NOS2CCNK
SCHEMBL2048413 0.87 MAPK14 (0.46) MAPK14NOS3NOS1NOS2CCNK
SCHEMBL16754485 0.87 MAPK14 (0.46) MAPK14NOS3NOS1NOS2CCNK
SCHEMBL16754749 0.87 MAPK14 (0.46) MAPK14NOS3NOS1NOS2CCNK
SCHEMBL17778616 0.81 ALDH1A1 (0.36) MAPK14CCNKCDK12KDM4EMEN1
SCHEMBL17778326 0.81 ALDH1A1 (0.36) MAPK14CCNKCDK12KDM4EMEN1
SCHEMBL12012111 0.80 NFE2L2 (0.47) MAPK14CA2
SCHEMBL17778156 0.80 ALDH1A1 (0.35) MAPK14CCNKCDK12KDM4EMEN1
SCHEMBL16775792 0.80 NOS3 (0.43) NOS3NOS1NOS2CCNKCDK12
SCHEMBL16775791 0.80 NOS3 (0.43) NOS3NOS1NOS2CCNKCDK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016079711-A1 SUBSTITUTED BRIDGED UREA ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-26 WO disclosed