SCHEMBL17791229

SCHEMBL17791229

C=CCn1cc(F)c(=O)[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.49
KDM4E B2RXH2 1/20 0.49
GRIA1 P42261 1/20 0.49
GRIA2 P42262 1/20 0.49
GRIA3 P42263 1/20 0.49
GRIA4 P48058 1/20 0.49
GRIK5 Q16478 1/20 0.49
LMNA P02545 2/20 0.47
KMT2A Q03164 2/20 0.47
CA12 O43570 7/20 0.39
CA9 Q16790 7/20 0.39
CA1 P00915 6/20 0.39
CA2 P00918 6/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TK1 P04183 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2559163 0.84 KDM4E (0.50) CYP1A2KDM4EGRIA1GRIA2GRIA3
SCHEMBL9891078 0.79 LMNA (0.51) CYP1A2KDM4EGRIA1GRIA2GRIA3
SCHEMBL14480450 0.79 KDM4E (0.47) CYP1A2KDM4EGRIA1GRIA2GRIA3
SCHEMBL148953 0.79 CYP3A4 (0.37) CYP1A2KDM4ELMNAKMT2ACYP3A4
SCHEMBL9021896 0.79 TK1 (0.56) TK1
SCHEMBL4564516 0.79 GRIA1 (0.49) CYP1A2GRIA1GRIA2GRIA4GRIK5
SCHEMBL17232952 0.78 LMNA (0.47) CYP1A2KDM4EGRIA1GRIA2GRIA3
SCHEMBL12410891 0.77 TK1 (0.41) CYP1A2KDM4EKMT2ACYP3A4CYP2D6
SCHEMBL11400618 0.77 KDM4E (0.54) CYP1A2KDM4EGRIA1GRIA2GRIA3
SCHEMBL1700458 0.76 LMNA (0.51) CYP1A2KDM4EGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160152573-A1 BIOORTHOGONAL METHODS AND COMPOUNDS THE UNIVERSITY COURT OF THE UNIVERSITY OF EDINBURGH (GB) 2016-06-02 US disclosed
US-20160152573-A1 BIOORTHOGONAL METHODS AND COMPOUNDS THE UNIVERSITY COURT OF THE UNIVERSITY OF EDINBURGH (GB) 2016-06-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160152573-A1 BIOORTHOGONAL METHODS AND COMPOUNDS DDT, DPYD, DNPEP CYP1A2 358/4885KDM4E 1986/4885GRIA1 3195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.