SCHEMBL17797443

SCHEMBL17797443

COC[C@@H](OC(N)=O)c1ccc(OC(F)(F)F)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 18/20 0.51
EPHX2 P34913 1/20 0.42
PDE1A P54750 1/20 0.41
PDE4D Q08499 1/20 0.41
SLC7A5 Q01650 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114750 1.00 PDE2A (0.51) PDE2AEPHX2PDE1APDE4DSLC7A5
SCHEMBL19946337 0.85 PDE2A (0.50) PDE2AEPHX2SLC7A5
SCHEMBL18045497 0.81 EPHX1 (0.43) PDE2AEPHX2SLC7A5
SCHEMBL28700452 0.79 TRPM8 (0.43) PDE2A
SCHEMBL28700451 0.79 TRPM8 (0.43) PDE2A
SCHEMBL19946332 0.78 PDE2A (0.53) PDE2AEPHX2SLC7A5
SCHEMBL18036164 0.78 PDE2A (0.59) PDE2AEPHX2PDE1APDE4DSLC7A5
SCHEMBL16563727 0.78 PDE2A (0.59) PDE2AEPHX2PDE1APDE4DSLC7A5
SCHEMBL19946338 0.78 PDE2A (0.64) PDE2AEPHX2
Hydrochloric Acid SCHEMBL16563850 0.77 PDE2A (0.58) PDE2AEPHX2PDE1APDE4DSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104245698-B Nitrogen-containing heterocyclic compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-11-30 CN disclosed
US-20160159808-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160159808-A1 HETEROCYCLIC COMPOUND PDE2A, PDE3A, PDE5A PDE2A 1/4885EPHX2 862/4885PDE1A 14/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.