SCHEMBL17801040

SCHEMBL17801040

N#Cc1ccc(-c2n[nH]c3ccc(-c4nnc(C5CCCN5)o4)cc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 1/20 0.51
TLR8 Q9NR97 1/20 0.51
TLR7 Q9NYK1 1/20 0.51
LRRK2 Q5S007 16/20 0.43
ITK Q08881 1/20 0.38
TRPA1 O75762 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17801034 0.78 LRRK2 (0.43) TLR9TLR8TLR7LRRK2ITK
SCHEMBL5384307 0.73 CYP2C19 (0.48) TLR9TLR8TLR7
SCHEMBL17801032 0.72 TLR8 (0.46) TLR9TLR8TLR7LRRK2ITK
SCHEMBL2636042 0.70 ALDH1A1 (0.61) TLR9TLR8TLR7
SCHEMBL16463738 0.70 CYP2C19 (0.55) TLR9TLR8TLR7
SCHEMBL16463737 0.70 CYP2C19 (0.55) TLR9TLR8TLR7
SCHEMBL19385363 0.69 USP30 (0.54) TLR9TLR8TLR7
SCHEMBL21065192 0.69 HPGD (0.51) TLR9TLR8TLR7
SCHEMBL13114282 0.69 ALDH1A1 (0.57) TLR9TLR8TLR7
SCHEMBL23115433 0.68 TLR8 (1.00) TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed