SCHEMBL17801100

SCHEMBL17801100

CC(C)(C)OC(=O)N1CCCC1c1n[nH]c(-c2ccc3[nH]nc(-c4cccc(NC(=O)C5CC5)c4)c3c2)n1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 6/20 0.44
PDPK1 O15530 2/20 0.43
CLK2 P49760 6/20 0.43
CLK3 P49761 6/20 0.43
DYRK1A Q13627 6/20 0.43
AAK1 Q2M2I8 2/20 0.42
ITK Q08881 2/20 0.41
SCN9A Q15858 1/20 0.40
TGFBR1 P36897 1/20 0.40
MAP3K5 Q99683 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17801042 0.81 CHEK2 (0.39) PDPK1
SCHEMBL17801079 0.79 PDPK1 (0.49) WNT1PDPK1CLK2CLK3DYRK1A
SCHEMBL2865036 0.74 PDPK1 (0.65) PDPK1AAK1ITK
SCHEMBL17801054 0.73 CPT1A (0.55) MAP3K5
SCHEMBL17801010 0.73 HCRTR2 (0.44)
SCHEMBL17801046 0.72 CPT1A (0.45) PDPK1MAP3K5
SCHEMBL5381303 0.71 AAK1 (0.52) WNT1PDPK1CLK2CLK3DYRK1A
SCHEMBL5377953 0.70 CLK2 (0.53) WNT1PDPK1CLK2CLK3DYRK1A
SCHEMBL4917155 0.70 NPC1 (0.51)
SCHEMBL6786829 0.70 ROCK1 (0.62)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016089977-A1 SUBSTITUTED INDAZOLE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH CELGENE CORPORATION (US) 2016-06-09 WO disclosed