SCHEMBL17802430

SCHEMBL17802430

O=C(O)c1ccc2ncc3cn[nH]c3c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
KDM4E B2RXH2 7/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
MGAM O43451 1/20 0.37
PLK4 O00444 1/20 0.36
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
DAPK3 O43293 1/20 0.36
MAP4K4 O95819 1/20 0.36
CSF1R P07333 1/20 0.36
RET P07949 1/20 0.36
FGFR1 P11362 1/20 0.36
PDGFRA P16234 1/20 0.36
LTK P29376 1/20 0.36
KDR P35968 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17802429 0.73 ALOX15 (0.39) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL30729983 0.72 TDP1 (0.41) ALDH1A1HPGDHSD17B10KDM4EKMT2A
SCHEMBL31721178 0.70 KDM4E (0.46) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL31721176 0.70 KDM4E (0.46) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL2022195 0.70 KDM4E (0.46) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL324668 0.69 KDM4E (0.47) ALOX15ALDH1A1HSD17B10KDM4ELMNA
SCHEMBL30483401 0.67 NAMPT (0.49) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL4994747 0.67 NAMPT (0.49) ALOX15ALDH1A1HPGDHSD17B10KDM4E
SCHEMBL7802908 0.67 ALDH1A1 (0.56) ALDH1A1HPGDHSD17B10KDM4EKMT2A
SCHEMBL13313392 0.66 KDM4E (0.46) ALOX15ALDH1A1HPGDHSD17B10KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3226862-A1 ORGANIC COMPOUNDS Intra-Cellular Therapies, Inc. (US) 2017-10-11 EP disclosed
WO-2016090382-A1 ORGANIC COMPOUNDS INTRA-CELLULAR THERAPIES, INC. (US) 2016-06-09 WO disclosed