SCHEMBL17804359

SCHEMBL17804359

CC(=O)c1cccc(N)c1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.44
ALDH1A1 P00352 7/20 0.42
HSD17B10 Q99714 6/20 0.42
CFTR P13569 1/20 0.42
BRD4 O60885 1/20 0.40
MAPT P10636 2/20 0.39
GAA P10253 1/20 0.39
KDM4E B2RXH2 6/20 0.38
HPGD P15428 4/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
FADS1 O60427 1/20 0.37
NSD2 O96028 2/20 0.37
TSHR P16473 2/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13468038 0.81 MMP2 (0.39) MMP2ALDH1A1HSD17B10CFTRMAPT
SCHEMBL5227176 0.81 MMP2 (0.61) MMP2ALDH1A1HSD17B10MAPTGAA
SCHEMBL29586692 0.81 MMP2 (0.61) MMP2ALDH1A1HSD17B10MAPTGAA
SCHEMBL11206826 0.79 PARP1 (0.44) ALDH1A1HSD17B10MAPTGAAKDM4E
SCHEMBL19972048 0.79 MMP2 (0.44) MMP2ALDH1A1HSD17B10CFTRMAPT
SCHEMBL5210612 0.79 ALDH1A1 (0.67) ALDH1A1HSD17B10CFTRMAPTGAA
SCHEMBL1873518 0.78 KMT2A (0.41) ALDH1A1HSD17B10KDM4EHPGDLMNA
SCHEMBL505381 0.78 MMP2 (0.47) MMP2ALDH1A1HSD17B10CFTRBRD4
2-Aminoacetophenone SCHEMBL29366456 0.78 ALDH1A1 (0.59) MMP2ALDH1A1HSD17B10CFTRBRD4
2-Aminoacetophenone SCHEMBL309044 0.78 ALDH1A1 (0.59) MMP2ALDH1A1HSD17B10CFTRBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3165520-A1 SUBSTITUTED BENZENE COMPOUNDS Epizyme Inc (US) 2017-05-10 EP disclosed
EP-2697198-B1 SUBSTITUTED BENZENE COMPOUNDS EPIZYME INC (US) 2016-06-08 EP disclosed
CN-1711247-A Celecoxib prodrug PHARMACIA CORP (US) 2005-12-21 CN disclosed