SCHEMBL178046

SCHEMBL178046

CC(Cc1ncc(-c2ccc(NC(=O)N3CCC(c4ccccc4)CC3)cc2)s1)C(C)(C)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 10/20 0.47
NPC1 O15118 6/20 0.46
RAB9A P51151 5/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
MAPT P10636 4/20 0.46
STAT1 P42224 1/20 0.46
TP53 P04637 4/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
MCHR1 Q99705 1/20 0.44
NFKB1 P19838 2/20 0.43
NFKB2 Q00653 2/20 0.43
RELA Q04206 2/20 0.43
LMNA P02545 1/20 0.43
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL178215 0.87 KDM4E (0.43) NAMPTKDM4E
SCHEMBL161913 0.85 NAMPT (0.47) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL178045 0.82 NAMPT (0.46) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL165730 0.81 NAMPT (0.45) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL27930087 0.80 OPRM1 (0.37) SMN1; SMN2CYP3A4HTT
SCHEMBL162335 0.72 RAB9A (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1HSD17B10
SCHEMBL159074 0.71 DGAT1 (0.42) SMN1; SMN2
SCHEMBL1172000 0.71 NPC1 (0.83) NAMPTNPC1RAB9ASMN1; SMN2MAPT
SCHEMBL162111 0.70 RAB9A (0.46) NPC1RAB9ASMN1; SMN2MAPTTP53
Hydrochloric Acid SCHEMBL161862 0.70 KDM4E (0.44) NAMPTSMN1; SMN2MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611783-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS Piramal Enterprises Limited (IN) 2013-07-10 EP disclosed
WO-2012029032-A2 HETEROCYCLIC COMPOUNDS AS DGAT1 INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2012-03-08 WO disclosed