SCHEMBL17819331

SCHEMBL17819331

Cc1c(-c2ccnn2-c2ccc(C#N)cc2)n(C(=O)NC2CCOC2)c(=O)n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ELANE P08246 19/20 0.54
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17819310 1.00 ELANE (0.54) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL17819338 1.00 ELANE (0.54) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL17861102 0.96 ELANE (0.55) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL17819351 0.93 ELANE (0.58) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL17819348 0.92 ELANE (0.57) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL17819344 0.92 ELANE (0.57) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL21859873 0.91 ELANE (0.56) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL19502788 0.90 ELANE (0.55) ELANEMEN1KMT2ACYP2C9CYP3A4
SCHEMBL21860404 0.89 ELANE (0.54) ELANEMEN1KMT2A
SCHEMBL21835826 0.89 ELANE (0.54) ELANEMEN1KMT2ACYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233833-B1 NOVEL COMPOUNDS CHIESI FARM SPA (IT) 2019-02-20 EP claimed
US-9409870-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2016-08-09 US claimed
US-20160168101-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2016-06-16 US claimed
EP-3464273-B9 IMIDAZOLONE COMPOUNDS AS HUMAN NEUTROPHIL ELASTASE INHIBITORS CHIESI FARM SPA (IT) 2020-10-21 EP disclosed
EP-3464273-B1 IMIDAZOLONE COMPOUNDS AS HUMAN NEUTROPHIL ELASTASE INHIBITORS CHIESI FARM SPA (IT) 2020-04-08 EP disclosed
EP-3464269-B1 HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF A HNE RELATED DISEASE CHIESI FARM SPA (IT) 2020-04-01 EP disclosed
EP-3233833-B1 NOVEL COMPOUNDS CHIESI FARM SPA (IT) 2019-02-20 EP disclosed
EP-3233833-B1 NOVEL COMPOUNDS CHIESI FARM SPA (IT) 2019-02-20 EP disclosed
US-10023558-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2018-07-17 US disclosed
US-20180009787-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2018-01-11 US disclosed
US-9862706-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2018-01-09 US disclosed
US-20170342056-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2017-11-30 US disclosed
US-9802919-B1 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2017-10-31 US disclosed
EP-3233833-A1 NOVEL COMPOUNDS Chiesi Farmaceutici S.p.A. (IT) 2017-10-25 EP disclosed
US-9409870-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2016-08-09 US disclosed
US-9409870-B2 Compounds CHIESI FARMACEUTICI S.P.A. (IT) 2016-08-09 US disclosed
WO-2016096638-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2016-06-23 WO disclosed
WO-2016096638-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2016-06-23 WO disclosed
US-20160168101-A1 NOVEL COMPOUNDS CHIESI FARMACEUTICI S.P.A. (IT) 2016-06-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10023558-B2 Compounds SERPINB1, ELANE, MPO ELANE 2/4885MEN1 3964/4885KMT2A 3935/4885
US-20180009787-A1 NOVEL COMPOUNDS SERPINB1, ELANE, MPO ELANE 2/4885MEN1 4581/4885KMT2A 4199/4885
US-20170342056-A1 NOVEL COMPOUNDS SERPINB1, ELANE, MPO ELANE 2/4885MEN1 4287/4885KMT2A 4376/4885
US-20160168101-A1 NOVEL COMPOUNDS ELANE, SERPINB1, MPO ELANE 1/4885MEN1 4140/4885KMT2A 4210/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.