SCHEMBL17825839

SCHEMBL17825839

O=C(Cc1ccccc1)Nn1ccnn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
GAA P10253 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
EPHX2 P34913 1/20 0.45
CYP19A1 P11511 1/20 0.44
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
ELOVL1 Q9BW60 1/20 0.43
CACNA1G O43497 1/20 0.43
CACNA1I Q9P0X4 1/20 0.43
POLB P06746 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HPGD P15428 1/20 0.43
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1259259 0.81 MEN1 (0.51) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL3936139 0.74 MEN1 (0.48) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL14833338 0.72 CYP19A1 (0.47) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL7468100 0.71 CYP19A1 (0.50) MEN1KMT2AALDH1A1MAPTCYP19A1
SCHEMBL7107935 0.71 ALDH1A1 (0.77) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL9563921 0.70 ALDH1A1 (0.75) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL29185687 0.70 MEN1 (0.50) MEN1KMT2AL3MBTL1HDAC8HDAC6
SCHEMBL28698664 0.69 MAPK1 (0.45) KMT2AL3MBTL1ALDH1A1CYP19A1SMN1; SMN2
SCHEMBL4338282 0.69 KDM4E (0.50) MEN1KMT2AGAAALDH1A1MAPT
SCHEMBL6470572 0.68 MEN1 (0.65) MEN1KMT2AHDAC8HDAC6GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113387894-B 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2023-02-24 CN claimed
CN-113387894-A 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-09-14 CN claimed
CN-113387894-B 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2023-02-24 CN disclosed
CN-113387894-A 1-N-benzene acetonitrile amido-triazole and pyrimidine derivative, preparation method and application thereof 首都医科大学脑重大疾病研究中心(北京脑重大疾病研究院) 2021-09-14 CN disclosed
EP-3229801-A1 FACTOR IXA INHIBITORS Merck Sharp & Dohme Corp. (US) 2017-10-18 EP disclosed
WO-2016094260-A1 FACTOR IXA INHIBITORS MERCK SHARP & DOHME CORP. (US) 2016-06-16 WO disclosed