SCHEMBL17826591

SCHEMBL17826591

COc1ccc(C(=O)NC(=S)Nc2ccc(NC(=O)CCCCN)cc2)cc1C(F)(F)F

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 17/20 0.80
SIRT2 Q8IXJ6 17/20 0.52
SIRT3 Q9NTG7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16229388 0.91 SIRT1 (0.81) SIRT1SIRT2
Hydrochloric Acid SCHEMBL1707264 0.83 SIRT1 (0.66) SIRT1
Hydrochloric Acid SCHEMBL1707261 0.83 SIRT1 (0.66) SIRT1
SCHEMBL17826589 0.82 SIRT1 (0.60) SIRT1SIRT2SIRT3
SCHEMBL17826586 0.81 SIRT2 (0.77) SIRT1SIRT2SIRT3
SCHEMBL14095986 0.80 SIRT1 (0.65) SIRT1SIRT2
SCHEMBL17826583 0.79 ALDH1A1 (0.64) SIRT1SIRT2
SCHEMBL14095988 0.79 SIRT1 (0.64) SIRT1
SCHEMBL17826579 0.79 SIRT2 (0.63) SIRT1SIRT2SIRT3
SCHEMBL17826590 0.78 SIRT2 (0.66) SIRT1SIRT2SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9365508-B2 Aroyl thiourea derivatives UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS (GB) 2016-06-14 US disclosed