SCHEMBL17826997

SCHEMBL17826997

CCc1cc(CN2CCN(C(=O)OC(C)(C)C)CC2)c2ccccc2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.50
CHRM4 P08173 1/20 0.50
CHRM1 P11229 1/20 0.50
CHRM3 P20309 1/20 0.50
GBA1 P04062 2/20 0.47
ADAM17 P78536 1/20 0.47
ACKR3 P25106 3/20 0.46
CKS1B P61024 1/20 0.45
SKP1 P63208 1/20 0.45
SKP2 Q13309 1/20 0.45
KMT2A Q03164 1/20 0.44
NSD2 O96028 1/20 0.44
IDO1 P14902 1/20 0.44
TDO2 P48775 1/20 0.44
IDO2 Q6ZQW0 1/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
VEGFA P15692 1/20 0.43
EGLN1 Q9GZT9 1/20 0.43
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17447752 0.86 CHRM2 (0.51) CHRM2CHRM4CHRM1CHRM3GBA1
SCHEMBL24696026 0.82 CHRM2 (0.47) CHRM2CHRM4CHRM1CHRM3GBA1
SCHEMBL16855926 0.81 FAAH (0.60) CHRM2CHRM4CHRM1CHRM3ACKR3
SCHEMBL3709871 0.80 FAAH (0.60) CHRM2CHRM4CHRM1CHRM3GBA1
SCHEMBL16830462 0.78 ACHE (0.60) CHRM2CHRM4CHRM1CHRM3KMT2A
SCHEMBL30422174 0.78 ACHE (0.60) CHRM2CHRM4CHRM1CHRM3KMT2A
SCHEMBL23293544 0.78 ACHE (0.60) CHRM2CHRM4CHRM1CHRM3KMT2A
SCHEMBL30958238 0.78 CHRM2 (0.52) CHRM2CHRM4CHRM1CHRM3GBA1
SCHEMBL19475343 0.78 MOK (0.72)
SCHEMBL29111354 0.77 GAA (0.66) ALDH1A1KDM4ETSHRNPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2152692-B1 COMPOUNDS WITH ANTI-CANCER ACTIVITY CANBAS CO LTD (JP) 2016-06-15 EP disclosed