SCHEMBL17834839

SCHEMBL17834839

Cc1csc2c(Br)nc(Br)cc12

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.33
CYP2A6 P11509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29959330 1.00 KCNA3 (0.33) KCNA3CYP2A6
SCHEMBL17822179 0.71 PIK3CA (0.47)
SCHEMBL25822955 0.69 CCR1 (0.33) CYP2A6
SCHEMBL25822909 0.65 CYP2A6 (0.43) CYP2A6
SCHEMBL23218344 0.65 CYP2A6 (0.32) KCNA3CYP2A6
SCHEMBL4264988 0.65 CYP2A6 (0.47) KCNA3CYP2A6
SCHEMBL12137043 0.63 GPR35 (0.32) CYP2A6
SCHEMBL11985866 0.63 TDP1 (0.35)
SCHEMBL19296324 0.63 CYP2A6 (0.32) CYP2A6
SCHEMBL4420462 0.62 CYP2A6 (0.41) KCNA3CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240199637-A1 IMPROVED PROCESS FOR THE PREPARATION OF 7-(MORPHOLINYL)-2-(N-PIPERAZINYL)METHYLTHIENO[2, 3-C]PYRIDINE DERIVATIVES NATCO PHARMA LIMITED (IN) 2024-06-20 US disclosed
EP-4326276-A1 IMPROVED PROCESS FOR THE PREPARATION OF 7-(MORPHOLINYL)-2-(N-PIPERAZINYL)METHYLTHIENO[2, 3-C]PYRIDINE DERIVATIVES Natco Pharma Ltd (IN) 2024-02-28 EP disclosed
CN-117529325-A Improved process for preparing 7- (morpholinyl) -2- (N-piperazinyl) methylthio [2,3-c ] pyridine derivatives 纳特科药品有限公司 2024-02-06 CN disclosed
CN-107074873-B 7- (morpholinyl) -2- (N-piperazinyl) methylthioeno [2, 3-c ] pyridine derivatives as anticancer agents 纳科法尔马有限公司 2022-01-07 CN disclosed
EP-3230289-B1 7-(MORPHOLINYL)-2-(N-PIPERAZINYL) METHYL THIENO [2, 3-C]PYRIDINE DERIVATIVES AS ANTICANCER DRUGS NATCO PHARMA LTD (IN) 2019-08-14 EP disclosed
US-20170320891-A1 7-(MORPHOLINYL)-2-(N-PIPERAZINYL) METHYL THIENO [2, 3-C] PYRIDINE DERIVATIVES AS ANTICANCER DRUGS NATCO PHARMA LIMITED (IN) 2017-11-09 US disclosed
US-20170320891-A1 7-(MORPHOLINYL)-2-(N-PIPERAZINYL) METHYL THIENO [2, 3-C] PYRIDINE DERIVATIVES AS ANTICANCER DRUGS NATCO PHARMA LIMITED (IN) 2017-11-09 US disclosed
WO-2016092556-A1 7-(MORPHOLINYL)-2-(N-PIPERAZINYL) METHYL THIENO [2, 3-C] PYRIDINE DERIVATIVES AS ANTICANCER DRUGS NATCO PHARMA LIMITED (IN) 2016-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240199637-A1 IMPROVED PROCESS FOR THE PREPARATION OF 7-(MORPHOLINYL)-2-(N-PIPERAZINYL)METHYLTHIENO[2, 3-C]PYRIDINE DERIVATIVES NR2C2, NRDC, NDC1 KCNA3 1667/4885CYP2A6 656/4885
US-20170320891-A1 7-(MORPHOLINYL)-2-(N-PIPERAZINYL) METHYL THIENO [2, 3-C] PYRIDINE DERIVATIVES AS ANTICANCER DRUGS PRMT7, CDK7, CASP7 KCNA3 2202/4885CYP2A6 1903/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.