SCHEMBL23218344

SCHEMBL23218344

Cc1csc2c(O)cc(Br)cc12

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.32
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRA2 P47869 1/20 0.30
GABRB2 P47870 1/20 0.30
GPR35 Q9HC97 2/20 0.30
KCNA3 P22001 1/20 0.30
LMNA P02545 1/20 0.30
PRNP P04156 1/20 0.30
HPGD P15428 1/20 0.30
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
NOD2 Q9HC29 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12137043 0.74 GPR35 (0.32) CYP2A6GPR35
SCHEMBL10729992 0.69 CYP2A6 (0.39) CYP2A6GPR35KCNA3HPGD
SCHEMBL10832904 0.68 TRPA1 (0.41) CYP2A6LMNAHPGDHTT
SCHEMBL25012039 0.66 CYP3A4 (0.45) GABRA1GABRB1GABRA2GABRB2LMNA
SCHEMBL10859770 0.65 MEN1 (0.39) CYP2A6GPR35HPGD
SCHEMBL3483833 0.65 ESR1 (0.34) CYP2A6GPR35KCNA3LMNA
SCHEMBL3483971 0.65 CYP3A4 (0.40) CYP2A6GPR35KCNA3LMNAHPGD
SCHEMBL26204561 0.65 NMT1 (0.31) GPR35
SCHEMBL17834839 0.65 KCNA3 (0.33) CYP2A6KCNA3
SCHEMBL4264988 0.65 CYP2A6 (0.47) CYP2A6GPR35KCNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12558341-B2 Oral complement factor D inhibitors BIOCRYST PHARMACEUTICALS, INC. (US) 2026-02-24 US disclosed
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS WILMINGTON TRUST, NATIONAL ASSOCIATION 2025-06-12 US disclosed
EP-4041238-A1 ORAL COMPLEMENT FACTOR D INHIBITORS Biocryst Pharmaceuticals, Inc. (US) 2022-08-17 EP disclosed
CN-114502168-A Oral complement factor D inhibitors 拜奥克里斯特制药公司 2022-05-13 CN disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed
WO-2021072198-A1 ORAL COMPLEMENT FACTOR D INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2021-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12558341-B2 Oral complement factor D inhibitors CFD, CFH, CFB CYP2A6 1256/4885GABRA1 3792/4885GABRB1 3695/4885
US-20250186391-A1 ORAL COMPLEMENT FACTOR D INHIBITORS CFD, CFH, CFB CYP2A6 1436/4885GABRA1 4487/4885GABRB1 4598/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.