SCHEMBL17834843

SCHEMBL17834843

Cc1cc(-c2ccc(-c3cnc(-c4ccc(C[C@H](NC(=O)c5ccc(C(C)(C)C)s5)C(=O)N[C@H](C)C(=O)O)cc4)nc3)c(F)c2)ccc1OC(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIFC1 Q9BW19 8/20 0.34
ALOX5AP P20292 3/20 0.34
FEN1 P39748 3/20 0.34
MCL1 Q07820 1/20 0.33
FFAR1 O14842 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
KIF11 P52732 1/20 0.33
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
ITGB7 P26010 1/20 0.32
PRSS1 P07477 1/20 0.32
TMPRSS15 P98073 1/20 0.32
KLKB1 P03952 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32
CTSL P07711 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
SDCBP O00560 1/20 0.32
SDC2 P34741 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17834619 0.91 KLKB1 (0.39) KIFC1ALOX5APFEN1KIF11ITGB1
SCHEMBL17834620 0.89 KIFC1 (0.37) KIFC1ALOX5APFEN1MCL1SDCBP
SCHEMBL17834504 0.89 MME (0.41) KIFC1ALOX5APFEN1MCL1SDCBP
SCHEMBL17834840 0.88 ALOX5AP (0.42) KIFC1ALOX5APFEN1MCL1
SCHEMBL17834550 0.88 KIFC1 (0.36) KIFC1ALOX5APFEN1ITGB1SDCBP
SCHEMBL17834625 0.88 KIFC1 (0.37) KIFC1ALOX5APFEN1SDCBPSDC2
SCHEMBL17834905 0.88 SDCBP (0.40) KIFC1ALOX5APFEN1SDCBPSDC2
SCHEMBL17834439 0.87 MMP12 (0.37) KIFC1ALOX5APFEN1FFAR1FFAR4
SCHEMBL17834655 0.87 PRSS1 (0.34) KIFC1ALOX5APFEN1KIF11ITGB1
SCHEMBL17834494 0.87 KIFC1 (0.41) KIFC1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3230276-B1 GLP-1 RECEPTOR MODULATORS CELGENE INT II SARL (CH) 2020-09-02 EP disclosed
US-10034886-B2 GLP-1 receptor modulators CELGENE INTERNATIONAL II SÀRL (CH) 2018-07-31 US disclosed
US-20180021346-A1 NOVEL GLP-1 RECEPTOR MODULATORS RECEPTOS LLC 2018-01-25 US disclosed
US-9795613-B2 GLP-1 receptor modulators CELGENE INTERNATIONAL II SÀRL (CH) 2017-10-24 US disclosed
US-20160228450-A1 NOVEL GLP-1 RECEPTOR MODULATORS RECEPTOS LLC 2016-08-11 US disclosed
WO-2016094729-A1 GLP-1 RECEPTOR MODULATORS CELGENE INTERNATIONAL II SARL (CH) 2016-06-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160228450-A1 NOVEL GLP-1 RECEPTOR MODULATORS GLP1R, GIPR, NPY1R KIFC1 4738/4885ALOX5AP 3115/4885FEN1 3722/4885
US-20180021346-A1 NOVEL GLP-1 RECEPTOR MODULATORS GLP1R, GIPR, NPY1R KIFC1 4738/4885ALOX5AP 3115/4885FEN1 3722/4885
US-10034886-B2 GLP-1 receptor modulators GLP1R, GIPR, GCGR KIFC1 4749/4885ALOX5AP 3438/4885FEN1 3634/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.